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Synthesis and antiviral evaluation of cytisine derivatives against dengue virus types 1 and 2.
Bioorg Med Chem Lett. 2021 Dec 15;54:128437. doi: 10.1016/j.bmcl.2021.128437. Epub 2021 Nov 2.
Bioorg Med Chem Lett. 2021.
PMID: 34737087
Thionation of quinolizidine alkaloids and their derivatives via Lawesson's reagent.
Koval'skaya AV, Petrova PR, Tsypyshev DO, Lobov AN, Tsypysheva IP.
Koval'skaya AV, et al. Among authors: tsypyshev do.
Nat Prod Res. 2022 Jul;36(14):3538-3543. doi: 10.1080/14786419.2020.1868460. Epub 2021 Jan 4.
Nat Prod Res. 2022.
PMID: 33397149
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Involvement of Chaperone Sigma1R in the Anxiolytic Effect of Fabomotizole.
Voronin MV, Vakhitova YV, Tsypysheva IP, Tsypyshev DO, Rybina IV, Kurbanov RD, Abramova EV, Seredenin SB.
Voronin MV, et al. Among authors: tsypyshev do.
Int J Mol Sci. 2021 May 21;22(11):5455. doi: 10.3390/ijms22115455.
Int J Mol Sci. 2021.
PMID: 34064275
Free PMC article.
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Novel Multitarget Hydroxamic Acids with a Natural Origin CAP Group against Alzheimer's Disease: Synthesis, Docking and Biological Evaluation.
Neganova M, Aleksandrova Y, Suslov E, Mozhaitsev E, Munkuev A, Tsypyshev D, Chicheva M, Rogachev A, Sukocheva O, Volcho K, Klochkov S.
Neganova M, et al.
Pharmaceutics. 2021 Nov 8;13(11):1893. doi: 10.3390/pharmaceutics13111893.
Pharmaceutics. 2021.
PMID: 34834312
Free PMC article.
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Inhibition of dengue viruses by N-methylcytisine thio derivatives through targeting viral envelope protein and NS2B-NS3 protease.
Lin CS, Lu CH, Lin TH, Kiu YT, Kan JY, Chang YJ, Hung PY, Koval'skaya AV, Tsypyshev DO, Tsypysheva IP, Lin CW.
Lin CS, et al. Among authors: tsypyshev do.
Bioorg Med Chem Lett. 2024 Feb 1;99:129623. doi: 10.1016/j.bmcl.2024.129623. Epub 2024 Jan 18.
Bioorg Med Chem Lett. 2024.
PMID: 38242331
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Antiviral activity of amides and carboxamides of quinolizidine alkaloid (-)-cytisine against human influenza virus A (H1N1) and parainfluenza virus type 3.
Fedorova VA, Kadyrova RA, Slita AV, Muryleva AA, Petrova PR, Kovalskaya AV, Lobov AN, Zileeva ZR, Tsypyshev DO, Borisevich SS, Tsypysheva IP, Vakhitova JV, Zarubaev VV.
Fedorova VA, et al. Among authors: tsypyshev do.
Nat Prod Res. 2021 Nov;35(22):4256-4264. doi: 10.1080/14786419.2019.1696791. Epub 2019 Dec 2.
Nat Prod Res. 2021.
PMID: 31790286
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