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Acridine-O6-benzylguanine hybrids: Synthesis, DNA binding, MGMT inhibition and antiproliferative activity.
Eur J Med Chem. 2022 Jan 5;227:113909. doi: 10.1016/j.ejmech.2021.113909. Epub 2021 Oct 9.
Eur J Med Chem. 2022.
PMID: 34731767
Free article.
Harnessing an emissive guanine surrogate to design small-molecule fluorescent chemosensors of O6-methylguanine-DNA-methyltransferase (MGMT).
Fillion A, Franco Pinto J, Granzhan A.
Fillion A, et al. Among authors: franco pinto j.
Org Biomol Chem. 2022 Mar 2;20(9):1888-1892. doi: 10.1039/d2ob00208f.
Org Biomol Chem. 2022.
PMID: 35174383
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Optimization of G-Quadruplex Ligands through a SAR Study Combining Parallel Synthesis and Screening of Cationic Bis(acylhydrazones).
Reznichenko O, Leclercq D, Franco Pinto J, Mouawad L, Gabelica V, Granzhan A.
Reznichenko O, et al. Among authors: franco pinto j.
Chemistry. 2023 Jan 18;29(4):e202202427. doi: 10.1002/chem.202202427. Epub 2022 Nov 30.
Chemistry. 2023.
PMID: 36286608
Free PMC article.
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