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Synthesis and Pharmacological Evaluation of Novel 2,3,4,5-tetrahydro[1,3]diazepino[1,2-a]benzimidazole Derivatives as Promising Anxiolytic and Analgesic Agents.
Molecules. 2021 Oct 6;26(19):6049. doi: 10.3390/molecules26196049.
Molecules. 2021.
PMID: 34641593
Free PMC article.
Searching for new anxiolytic agents among derivatives of 11-dialkylaminoethyl-2,3,4,5-tetrahydrodiazepino[1,2-a]benzimidazole.
Maltsev DV, Spasov AA, Yakovlev DS, Vassiliev PM, Skripka MO, Miroshnikov MV, Sultanova KT, Kochetkov AN, Divaeva LN, Kuzmenko TA, Morkovnik AS.
Maltsev DV, et al. Among authors: miroshnikov mv.
Eur J Pharm Sci. 2021 Jun 1;161:105792. doi: 10.1016/j.ejps.2021.105792. Epub 2021 Mar 8.
Eur J Pharm Sci. 2021.
PMID: 33705965
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Synthesis and multifaceted pharmacological activity of novel quinazoline NHE-1 inhibitors.
Spasov A, Ozerov A, Vassiliev P, Kosolapov V, Gurova N, Kucheryavenko A, Naumenko L, Babkov D, Sirotenko V, Taran A, Litvinov R, Borisov A, Klochkov V, Merezhkina D, Miroshnikov M, Uskov G, Ovsyankina N.
Spasov A, et al.
Sci Rep. 2021 Dec 21;11(1):24380. doi: 10.1038/s41598-021-03722-w.
Sci Rep. 2021.
PMID: 34934125
Free PMC article.
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Discovery of Nitro-azolo[1,5-a]pyrimidines with Anti-Inflammatory and Protective Activity against LPS-Induced Acute Lung Injury.
Spasov A, Kosolapov V, Babkov D, Klochkov V, Sokolova E, Miroshnikov M, Borisov A, Velikorodnaya Y, Smirnov A, Savateev K, Fedotov V, Kotovskaya S, Rusinov V.
Spasov A, et al.
Pharmaceuticals (Basel). 2022 Apr 27;15(5):537. doi: 10.3390/ph15050537.
Pharmaceuticals (Basel). 2022.
PMID: 35631365
Free PMC article.
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Design, Synthesis and Pharmacological Evaluation of Novel C2,C3-Quinoxaline Derivatives as Promising Anxiolytic Agents.
Maltsev DV, Skripka MO, Spasov AA, Vassiliev PM, Perfiliev MA, Divaeva LN, Zubenko AA, Morkovnik AS, Klimenko AI, Miroshnikov MV, Klochkov VG, Ianalieva LR.
Maltsev DV, et al. Among authors: miroshnikov mv.
Int J Mol Sci. 2022 Nov 19;23(22):14401. doi: 10.3390/ijms232214401.
Int J Mol Sci. 2022.
PMID: 36430878
Free PMC article.
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Guanidine Derivatives of Quinazoline-2,4(1H,3H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents.
Spasov A, Ozerov A, Kosolapov V, Gurova N, Kucheryavenko A, Naumenko L, Babkov D, Sirotenko V, Taran A, Borisov A, Sokolova E, Klochkov V, Merezhkina D, Miroshnikov M, Ovsyankina N, Smirnov A, Velikorodnaya Y.
Spasov A, et al.
Life (Basel). 2022 Oct 20;12(10):1647. doi: 10.3390/life12101647.
Life (Basel). 2022.
PMID: 36295082
Free PMC article.
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