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Synthesis and Pharmacological Evaluation of Novel 2,3,4,5-tetrahydro[1,3]diazepino[1,2-a]benzimidazole Derivatives as Promising Anxiolytic and Analgesic Agents.
Molecules. 2021 Oct 6;26(19):6049. doi: 10.3390/molecules26196049.
Molecules. 2021.
PMID: 34641593
Free PMC article.
[Neural network modeling of multitarget RAGE inhibitory activity].
Vassiliev PM, Spasov AA, Yanaliyeva LR, Kochetkov AN, Vorfolomeyeva VV, Klochkov VG, Appazova DT.
Vassiliev PM, et al. Among authors: kochetkov an.
Biomed Khim. 2019 Feb;65(2):91-98. doi: 10.18097/PBMC20196502091.
Biomed Khim. 2019.
PMID: 30950813
Russian.
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Bornyl Derivatives of p-(Benzyloxy)Phenylpropionic Acid: In Vivo Evaluation of Antidiabetic Activity.
Kuranov S, Luzina O, Khvostov M, Baev D, Kuznetsova D, Zhukova N, Vassiliev P, Kochetkov A, Tolstikova T, Salakhutdinov N.
Kuranov S, et al.
Pharmaceuticals (Basel). 2020 Nov 19;13(11):404. doi: 10.3390/ph13110404.
Pharmaceuticals (Basel). 2020.
PMID: 33228030
Free PMC article.
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Searching for new anxiolytic agents among derivatives of 11-dialkylaminoethyl-2,3,4,5-tetrahydrodiazepino[1,2-a]benzimidazole.
Maltsev DV, Spasov AA, Yakovlev DS, Vassiliev PM, Skripka MO, Miroshnikov MV, Sultanova KT, Kochetkov AN, Divaeva LN, Kuzmenko TA, Morkovnik AS.
Maltsev DV, et al. Among authors: kochetkov an.
Eur J Pharm Sci. 2021 Jun 1;161:105792. doi: 10.1016/j.ejps.2021.105792. Epub 2021 Mar 8.
Eur J Pharm Sci. 2021.
PMID: 33705965
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[Consensus ensemble neural network multitarget model of RAGE inhibitory activity of chemical compounds].
Vassiliev PM, Spasov AA, Kochetkov AN, Perfilev MA, Koroleva AR.
Vassiliev PM, et al. Among authors: kochetkov an.
Biomed Khim. 2021 May;67(3):268-277. doi: 10.18097/PBMC20216703268.
Biomed Khim. 2021.
PMID: 34142534
Russian.
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Combined In Silico, Ex Vivo, and In Vivo Assessment of L-17, a Thiadiazine Derivative with Putative Neuro- and Cardioprotective and Antidepressant Effects.
Sarapultsev A, Vassiliev P, Grinchii D, Kiss A, Mach M, Osacka J, Balloova A, Paliokha R, Kochetkov A, Sidorova L, Sarapultsev P, Chupakhin O, Rantsev M, Spasov A, Dremencov E.
Sarapultsev A, et al.
Int J Mol Sci. 2021 Dec 20;22(24):13626. doi: 10.3390/ijms222413626.
Int J Mol Sci. 2021.
PMID: 34948423
Free PMC article.
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Consensus Ensemble Multitarget Neural Network Model of Anxiolytic Activity of Chemical Compounds and Its Use for Multitarget Pharmacophore Design.
Vassiliev PM, Maltsev DV, Spasov AA, Perfilev MA, Skripka MO, Kochetkov AN.
Vassiliev PM, et al. Among authors: kochetkov an.
Pharmaceuticals (Basel). 2023 May 11;16(5):731. doi: 10.3390/ph16050731.
Pharmaceuticals (Basel). 2023.
PMID: 37242513
Free PMC article.
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