Semysinthetic biflavonoid Morelloflavone-7,4',7″,3‴,4‴-penta-O-butanoyl is a more potent inhibitor of Proprotein Convertases Subtilisin/Kexin PC1/3 than Kex2 and Furin.
de Souza AA, de Andrade DM, Siqueira FDS, Di Iorio JF, Veloso MP, Coelho CM, Viegas Junior C, Gontijo VS, Dos Santos MH, Meneghetti MCZ, Nader HB, Tersariol ILDS, Juliano L, Juliano MA, Judice WAS.
de Souza AA, et al. Among authors: juliano l, juliano ma.
Biochim Biophys Acta Gen Subj. 2021 Dec;1865(12):130016. doi: 10.1016/j.bbagen.2021.130016. Epub 2021 Sep 22.
Biochim Biophys Acta Gen Subj. 2021.
PMID: 34560176