Karnik KS - Search Results

1

Free energy perturbation guided Synthesis with Biological Evaluation of Substituted Quinoline derivatives as small molecule L858R/T790M/C797S mutant EGFR inhibitors targeting resistance in Non-Small Cell Lung Cancer (NSCLC).

Karnik KS, Sarkate AP, Tiwari SV, Azad R, Wakte PS. Karnik KS, et al. Bioorg Chem. 2021 Oct;115:105226. doi: 10.1016/j.bioorg.2021.105226. Epub 2021 Jul 31. Bioorg Chem. 2021. PMID: 34364055

2

Synthesis and antimicrobial evaluation of novel ethyl 2-(2-(4-substituted)acetamido)-4-subtituted-thiazole-5-carboxylate derivatives.

Pawar CD, Sarkate AP, Karnik KS, Bahekar SS, Pansare DN, Shelke RN, Jawale CS, Shinde DB. Pawar CD, et al. Among authors: karnik ks. Bioorg Med Chem Lett. 2016 Aug 1;26(15):3525-8. doi: 10.1016/j.bmcl.2016.06.030. Epub 2016 Jun 11. Bioorg Med Chem Lett. 2016. PMID: 27324976

3

Development of triple mutant T790M/C797S allosteric EGFR inhibitors: a computational approach.

Karnik KS, Sarkate AP, Lokwani DK, Narula IS, Burra PVLS, Wakte PS. Karnik KS, et al. J Biomol Struct Dyn. 2021 Sep;39(15):5376-5398. doi: 10.1080/07391102.2020.1786460. Epub 2020 Jul 1. J Biomol Struct Dyn. 2021. PMID: 32608331

4

Ultrasound assisted synthesis of tetrazole based pyrazolines and isoxazolines as potent anticancer agents via inhibition of tubulin polymerization.

Dofe VS, Sarkate AP, Tiwari SV, Lokwani DK, Karnik KS, Kale IA, Dodamani S, Jalalpure SS, Burra PVLS. Dofe VS, et al. Among authors: karnik ks. Bioorg Med Chem Lett. 2020 Nov 15;30(22):127592. doi: 10.1016/j.bmcl.2020.127592. Epub 2020 Sep 30. Bioorg Med Chem Lett. 2020. PMID: 33010448

5

Computational and Synthetic approach with Biological Evaluation of Substituted Quinoline derivatives as small molecule L858R/T790M/C797S triple mutant EGFR inhibitors targeting resistance in Non-Small Cell Lung Cancer (NSCLC).

Karnik KS, Sarkate AP, Tiwari SV, Azad R, Burra PVLS, Wakte PS. Karnik KS, et al. Bioorg Chem. 2021 Feb;107:104612. doi: 10.1016/j.bioorg.2020.104612. Epub 2021 Jan 5. Bioorg Chem. 2021. PMID: 33476869

6

One pot synthesis, in silico study and evaluation of some novel flavonoids as potent topoisomerase II inhibitors.

Sarkate AP, Dofe VS, Tiwari SV, Lokwani DK, Karnik KS, Kamble DD, Ansari MHSH, Dodamani S, Jalalpure SS, Sangshetti JN, Azad R, Burra PVLS, Bhandari SV. Sarkate AP, et al. Among authors: karnik ks. Bioorg Med Chem Lett. 2021 May 15;40:127916. doi: 10.1016/j.bmcl.2021.127916. Epub 2021 Mar 6. Bioorg Med Chem Lett. 2021. PMID: 33689875

7

Molecular dynamic simulations based discovery and development of thiazolidin-4-one derivatives as EGFR inhibitors targeting resistance in non-small cell lung cancer (NSCLC).

Karnik KS, Sarkate AP, Lokwani DK, Tiwari SV, Azad R, Wakte PS. Karnik KS, et al. J Biomol Struct Dyn. 2023 Jul;41(10):4696-4710. doi: 10.1080/07391102.2022.2071339. Epub 2022 May 9. J Biomol Struct Dyn. 2023. PMID: 35532095

8

Facile Synthesis of Novel Coumarin Derivatives, Antimicrobial Analysis, Enzyme Assay, Docking Study, ADMET Prediction and Toxicity Study.

Tiwari SV, Seijas JA, Vazquez-Tato MP, Sarkate AP, Karnik KS, Nikalje APG. Tiwari SV, et al. Among authors: karnik ks. Molecules. 2017 Jul 13;22(7):1172. doi: 10.3390/molecules22071172. Molecules. 2017. PMID: 28703783 Free PMC article.

9

Novel 2-(nitrooxy)ethyl 2-(4-(substituted phenyl)-2-((substituted phenyl)amino)thiazol-5-yl)acetate as Anti-inflammatory, Analgesic and Nitric Oxide Releasing Agents: Synthesis and Molecular Docking Studies.

Sarkate AP, Lokwani DK, Karnik KS, Shinde DB. Sarkate AP, et al. Among authors: karnik ks. Antiinflamm Antiallergy Agents Med Chem. 2017;16(3):153-167. doi: 10.2174/1871523016666171115125922. Antiinflamm Antiallergy Agents Med Chem. 2017. PMID: 29141568

10

Ionic Liquid-Promoted Synthesis of Novel Chromone-Pyrimidine Coupled Derivatives, Antimicrobial Analysis, Enzyme Assay, Docking Study and Toxicity Study.

Tiwari SV, Seijas JA, Vazquez-Tato MP, Sarkate AP, Karnik KS, Nikalje APG. Tiwari SV, et al. Among authors: karnik ks. Molecules. 2018 Feb 16;23(2):440. doi: 10.3390/molecules23020440. Molecules. 2018. PMID: 29462951 Free PMC article.

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