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3CL Protease Inhibitors with an Electrophilic Arylketone Moiety as Anti-SARS-CoV-2 Agents.
Konno S, Kobayashi K, Senda M, Funai Y, Seki Y, Tamai I, Schäkel L, Sakata K, Pillaiyar T, Taguchi A, Taniguchi A, Gütschow M, Müller CE, Takeuchi K, Hirohama M, Kawaguchi A, Kojima M, Senda T, Shirasaka Y, Kamitani W, Hayashi Y. Konno S, et al. J Med Chem. 2022 Feb 24;65(4):2926-2939. doi: 10.1021/acs.jmedchem.1c00665. Epub 2021 Jul 27. J Med Chem. 2022. PMID: 34313428
Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: structure-activity relationship study.
Thanigaimalai P, Konno S, Yamamoto T, Koiwai Y, Taguchi A, Takayama K, Yakushiji F, Akaji K, Kiso Y, Kawasaki Y, Chen SE, Naser-Tavakolian A, Schön A, Freire E, Hayashi Y. Thanigaimalai P, et al. Among authors: konno s. Eur J Med Chem. 2013 Jul;65:436-47. doi: 10.1016/j.ejmech.2013.05.005. Epub 2013 May 20. Eur J Med Chem. 2013. PMID: 23747811 Free PMC article.
Development of potent dipeptide-type SARS-CoV 3CL protease inhibitors with novel P3 scaffolds: design, synthesis, biological evaluation, and docking studies.
Thanigaimalai P, Konno S, Yamamoto T, Koiwai Y, Taguchi A, Takayama K, Yakushiji F, Akaji K, Chen SE, Naser-Tavakolian A, Schön A, Freire E, Hayashi Y. Thanigaimalai P, et al. Among authors: konno s. Eur J Med Chem. 2013 Oct;68:372-84. doi: 10.1016/j.ejmech.2013.07.037. Epub 2013 Aug 9. Eur J Med Chem. 2013. PMID: 23994330 Free PMC article.
Structural Revision of Natural Cyclic Depsipeptide MA026 Established by Total Synthesis and Biosynthetic Gene Cluster Analysis.
Uchiyama C, Fukuda A, Mukaiyama M, Nakazawa Y, Kuramochi Y, Muguruma K, Arimoto M, Ninomiya A, Kako K, Katsuyama Y, Konno S, Taguchi A, Takayama K, Taniguchi A, Nagumo Y, Usui T, Hayashi Y. Uchiyama C, et al. Among authors: konno s. Angew Chem Int Ed Engl. 2021 Apr 12;60(16):8792-8797. doi: 10.1002/anie.202015193. Epub 2021 Mar 8. Angew Chem Int Ed Engl. 2021. PMID: 33533101
Inactivation of myostatin by photooxygenation using functionalized d-peptides.
Okamoto H, Murano SA, Ikekawa K, Katsuyama M, Konno S, Taguchi A, Takayama K, Taniguchi A, Hayashi Y. Okamoto H, et al. Among authors: konno s. RSC Med Chem. 2023 Jan 3;14(2):386-392. doi: 10.1039/d2md00425a. eCollection 2023 Feb 22. RSC Med Chem. 2023. PMID: 36846372 Free PMC article.
X-Ray Conformation and Structure-Activity Relationships of MA026, a Reversible Tight Junction Opener.
Mukaiyama M, Uchiyama C, Fukuda A, Nakazawa Y, Kuramochi Y, Shibata Y, Konno S, Muguruma K, Matsugaki N, Asari T, Ogawa K, Taguchi A, Takayama K, Taniguchi A, Nagumo Y, Senda T, Hayashi Y, Usui T. Mukaiyama M, et al. Among authors: konno s. J Med Chem. 2023 Jul 13;66(13):8717-8724. doi: 10.1021/acs.jmedchem.3c00365. Epub 2023 Jun 23. J Med Chem. 2023. PMID: 37352439
1,259 results