Dessoy MA - Search Results

1

Hit-to-lead optimization of a benzene sulfonamide series for potential antileishmanial agents.

Koovits PJ, Dessoy MA, Matheeussen A, Maes L, Caljon G, Ferreira LLG, Chelucci RC, Michelan-Duarte S, Andricopulo AD, Campbell S, Kratz JM, Mowbray CE, Dias LC. Koovits PJ, et al. Among authors: dessoy ma. RSC Med Chem. 2020 Aug 25;11(11):1267-1274. doi: 10.1039/d0md00165a. RSC Med Chem. 2020. PMID: 34085041 Free PMC article.

2

Synthesis, biological evaluation, and structure-activity relationships of potent noncovalent and nonpeptidic cruzain inhibitors as anti-Trypanosoma cruzi agents.

Ferreira RS, Dessoy MA, Pauli I, Souza ML, Krogh R, Sales AI, Oliva G, Dias LC, Andricopulo AD. Ferreira RS, et al. Among authors: dessoy ma. J Med Chem. 2014 Mar 27;57(6):2380-92. doi: 10.1021/jm401709b. Epub 2014 Mar 3. J Med Chem. 2014. PMID: 24533839 Free article.

3

Molecular modeling and structure-activity relationships for a series of benzimidazole derivatives as cruzain inhibitors.

Pauli I, Ferreira LG, de Souza ML, Oliva G, Ferreira RS, Dessoy MA, Slafer BW, Dias LC, Andricopulo AD. Pauli I, et al. Among authors: dessoy ma. Future Med Chem. 2017 May;9(7):641-657. doi: 10.4155/fmc-2016-0236. Epub 2017 May 16. Future Med Chem. 2017. PMID: 28509592

4

Benzimidazole inhibitors of the major cysteine protease of Trypanosoma brucei.

Pereira GA, Santos LH, Wang SC, Martins LC, Villela FS, Liao W, Dessoy MA, Dias LC, Andricopulo AD, Costa MA, Nagem RA, Caffrey CR, Liedl KR, Caffarena ER, Ferreira RS. Pereira GA, et al. Among authors: dessoy ma. Future Med Chem. 2019 Jul;11(13):1537-1551. doi: 10.4155/fmc-2018-0523. Future Med Chem. 2019. PMID: 31469332 Free PMC article.

5

Structure-activity relationship of 4-azaindole-2-piperidine derivatives as agents against Trypanosoma cruzi.

Koovits PJ, Dessoy MA, Matheeussen A, Maes L, Caljon G, Mowbray CE, Kratz JM, Dias LC. Koovits PJ, et al. Among authors: dessoy ma. Bioorg Med Chem Lett. 2020 Jan 1;30(1):126779. doi: 10.1016/j.bmcl.2019.126779. Epub 2019 Oct 31. Bioorg Med Chem Lett. 2020. PMID: 31706667 Free article.

6

Multiparameter Optimization of Trypanocidal Cruzain Inhibitors With In Vivo Activity and Favorable Pharmacokinetics.

Pauli I, Rezende CO Jr, Slafer BW, Dessoy MA, de Souza ML, Ferreira LLG, Adjanohun ALM, Ferreira RS, Magalhães LG, Krogh R, Michelan-Duarte S, Del Pintor RV, da Silva FBR, Cruz FC, Dias LC, Andricopulo AD. Pauli I, et al. Among authors: dessoy ma. Front Pharmacol. 2022 Jan 5;12:774069. doi: 10.3389/fphar.2021.774069. eCollection 2021. Front Pharmacol. 2022. PMID: 35069198 Free PMC article.

7

Synthesis and Anti-Trypanosoma cruzi Activity of 3-Cyanopyridine Derivatives.

Slafer BW, Dessoy MA, de Oliveira RG, Mollo MC, Lee E, Matheeussen A, Maes L, Caljon G, Ferreira LLG, Krogh R, Andricopulo AD, Cruz LR, Mowbray CE, Kratz JM, Dias LC. Slafer BW, et al. Among authors: dessoy ma. ACS Omega. 2024 May 13;9(20):22360-22370. doi: 10.1021/acsomega.4c01919. eCollection 2024 May 21. ACS Omega. 2024. PMID: 38799347 Free PMC article.

8

Analysis of cytokinin nucleotides by capillary zone electrophoresis with diode array and mass spectrometric detection in a recombinant enzyme in vitro reaction.

Béres T, Gemrotová M, Tarkowski P, Ganzera M, Maier V, Friedecký D, Dessoy MA, Wessjohann LA, Spíchal L, Strnad M, Doležal K. Béres T, et al. Among authors: dessoy ma. Anal Chim Acta. 2012 Nov 2;751:176-81. doi: 10.1016/j.aca.2012.08.049. Epub 2012 Sep 5. Anal Chim Acta. 2012. PMID: 23084068

9

In vitro and in vivo production of new aminocoumarins by a combined biochemical, genetic, and synthetic approach.

Galm U, Dessoy MA, Schmidt J, Wessjohann LA, Heide L. Galm U, et al. Among authors: dessoy ma. Chem Biol. 2004 Feb;11(2):173-83. doi: 10.1016/j.chembiol.2004.01.012. Chem Biol. 2004. PMID: 15123279

10

A proposed mechanism for the reductive ring opening of the cyclodiphosphate MEcPP, a crucial transformation in the new DXP/MEP pathway to isoprenoids based on modeling studies and feeding experiments.

Brandt W, Dessoy MA, Fulhorst M, Gao W, Zenk MH, Wessjohann LA. Brandt W, et al. Among authors: dessoy ma. Chembiochem. 2004 Mar 5;5(3):311-23. doi: 10.1002/cbic.200300743. Chembiochem. 2004. PMID: 14997523

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