Bermudez M - Search Results

1

Allosteric coupling and biased agonism in G protein-coupled receptors.

Bock A, Bermudez M. Bock A, et al. Among authors: bermudez m. FEBS J. 2021 Apr;288(8):2513-2528. doi: 10.1111/febs.15783. Epub 2021 Mar 5. FEBS J. 2021. PMID: 33621418 Free article. Review.

2

Ligand Binding Ensembles Determine Graded Agonist Efficacies at a G Protein-coupled Receptor.

Bock A, Bermudez M, Krebs F, Matera C, Chirinda B, Sydow D, Dallanoce C, Holzgrabe U, De Amici M, Lohse MJ, Wolber G, Mohr K. Bock A, et al. Among authors: bermudez m. J Biol Chem. 2016 Jul 29;291(31):16375-89. doi: 10.1074/jbc.M116.735431. Epub 2016 Jun 13. J Biol Chem. 2016. PMID: 27298318 Free PMC article.

3

Structural Characteristics of the Allosteric Binding Site Represent a Key to Subtype Selective Modulators of Muscarinic Acetylcholine Receptors.

Bermudez M, Rakers C, Wolber G. Bermudez M, et al. Mol Inform. 2015 Aug;34(8):526-30. doi: 10.1002/minf.201500025. Epub 2015 Jul 1. Mol Inform. 2015. PMID: 27490498

4

Ligand-Specific Restriction of Extracellular Conformational Dynamics Constrains Signaling of the M₂ Muscarinic Receptor.

Bermudez M, Bock A, Krebs F, Holzgrabe U, Mohr K, Lohse MJ, Wolber G. Bermudez M, et al. ACS Chem Biol. 2017 Jul 21;12(7):1743-1748. doi: 10.1021/acschembio.7b00275. Epub 2017 Jun 12. ACS Chem Biol. 2017. PMID: 28585805

5

A panoramic view on GPCRs: the 1st Berlin Symposium for Interdisciplinary GPCR research.

Bock A, Bermudez M. Bock A, et al. Among authors: bermudez m. Naunyn Schmiedebergs Arch Pharmacol. 2018 Jul;391(7):769-771. doi: 10.1007/s00210-018-1513-5. Epub 2018 May 21. Naunyn Schmiedebergs Arch Pharmacol. 2018. PMID: 29781045 No abstract available.

6

Strategies for the discovery of biased GPCR ligands.

Bermudez M, Nguyen TN, Omieczynski C, Wolber G. Bermudez M, et al. Drug Discov Today. 2019 Apr;24(4):1031-1037. doi: 10.1016/j.drudis.2019.02.010. Epub 2019 Mar 1. Drug Discov Today. 2019. PMID: 30831262 Review.

7

Does Divergent Binding Pocket Closure Drive Ligand Bias for Class A GPCRs?

Bermudez M, Bock A. Bermudez M, et al. Trends Pharmacol Sci. 2019 Apr;40(4):236-239. doi: 10.1016/j.tips.2019.02.005. Epub 2019 Mar 6. Trends Pharmacol Sci. 2019. PMID: 30852058 Review.

8

Ligand-Specific Allosteric Coupling Controls G-Protein-Coupled Receptor Signaling.

Holze J, Bermudez M, Pfeil EM, Kauk M, Bödefeld T, Irmen M, Matera C, Dallanoce C, De Amici M, Holzgrabe U, König GM, Tränkle C, Wolber G, Schrage R, Mohr K, Hoffmann C, Kostenis E, Bock A. Holze J, et al. Among authors: bermudez m. ACS Pharmacol Transl Sci. 2020 Sep 2;3(5):859-867. doi: 10.1021/acsptsci.0c00069. eCollection 2020 Oct 9. ACS Pharmacol Transl Sci. 2020. PMID: 33073186 Free PMC article.

9

The Role of Orthosteric Building Blocks of Bitopic Ligands for Muscarinic M1 Receptors.

Volpato D, Kauk M, Messerer R, Bermudez M, Wolber G, Bock A, Hoffmann C, Holzgrabe U. Volpato D, et al. Among authors: bermudez m. ACS Omega. 2020 Dec 1;5(49):31706-31715. doi: 10.1021/acsomega.0c04220. eCollection 2020 Dec 15. ACS Omega. 2020. PMID: 33344823 Free PMC article.

10

Biased Ligands Differentially Shape the Conformation of the Extracellular Loop Region in 5-HT_2B Receptors.

Denzinger K, Nguyen TN, Noonan T, Wolber G, Bermudez M. Denzinger K, et al. Among authors: bermudez m. Int J Mol Sci. 2020 Dec 20;21(24):9728. doi: 10.3390/ijms21249728. Int J Mol Sci. 2020. PMID: 33419260 Free PMC article.

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