Makadia P - Search Results

1

Discovery of a potent G-protein-coupled receptor 119 agonist for the treatment of type 2 diabetes.

Pola S, Shah SR, Pingali H, Zaware P, Thube B, Makadia P, Patel H, Bandyopadhyay D, Rath A, Giri S, Patel JH, Ranvir RK, Sundar SR, Patel H, Kumar J, Jain MR. Pola S, et al. Among authors: makadia p. Bioorg Med Chem. 2021 Apr 1;35:116071. doi: 10.1016/j.bmc.2021.116071. Epub 2021 Feb 13. Bioorg Med Chem. 2021. PMID: 33611013

2

Design and synthesis of novel oxazole containing 1,3-dioxane-2-carboxylic acid derivatives as PPAR alpha/gamma dual agonists.

Pingali H, Jain M, Shah S, Makadia P, Zaware P, Goel A, Patel M, Giri S, Patel H, Patel P. Pingali H, et al. Among authors: makadia p. Bioorg Med Chem. 2008 Aug 1;16(15):7117-27. doi: 10.1016/j.bmc.2008.06.050. Epub 2008 Jun 28. Bioorg Med Chem. 2008. PMID: 18625559

3

Discovery of a highly orally bioavailable c-5-[6-(4-Methanesulfonyloxyphenyl)hexyl]-2-methyl-1,3-dioxane-r-2-carboxylic acid as a potent hypoglycemic and hypolipidemic agent.

Pingali H, Jain M, Shah S, Basu S, Makadia P, Goswami A, Zaware P, Patil P, Godha A, Giri S, Goel A, Patel M, Patel H, Patel P. Pingali H, et al. Among authors: makadia p. Bioorg Med Chem Lett. 2008 Oct 15;18(20):5586-90. doi: 10.1016/j.bmcl.2008.08.112. Epub 2008 Sep 3. Bioorg Med Chem Lett. 2008. PMID: 18805005

4

Design and synthesis of novel bis-oximinoalkanoic acids as potent PPAR alpha agonists.

Pingali H, Jain M, Shah S, Zaware P, Makadia P, Pola S, Thube B, Patel D, Patil P, Priyadarshini P, Suthar D, Shah M, Giri S, Patel P. Pingali H, et al. Among authors: makadia p. Bioorg Med Chem Lett. 2010 Feb 1;20(3):1156-61. doi: 10.1016/j.bmcl.2009.12.022. Epub 2009 Dec 6. Bioorg Med Chem Lett. 2010. PMID: 20022492

5

Modulation of PPAR subtype selectivity. Part 2: Transforming PPARα/γ dual agonist into α selective PPAR agonist through bioisosteric modification.

Zaware P, Shah SR, Pingali H, Makadia P, Thube B, Pola S, Patel D, Priyadarshini P, Suthar D, Shah M, Jamili J, Sairam KV, Giri S, Patel L, Patel H, Sudani H, Patel H, Jain M, Patel P, Bahekar R. Zaware P, et al. Among authors: makadia p. Bioorg Med Chem Lett. 2011 Jan 15;21(2):628-32. doi: 10.1016/j.bmcl.2010.12.032. Epub 2010 Dec 10. Bioorg Med Chem Lett. 2011. PMID: 21195611

6

Effect of structurally constrained oxime-ether linker on PPAR subtype selectivity: Discovery of a novel and potent series of PPAR-pan agonists.

Makadia P, Shah SR, Pingali H, Zaware P, Patel D, Pola S, Thube B, Priyadarshini P, Suthar D, Shah M, Giri S, Trivedi C, Jain M, Patel P, Bahekar R. Makadia P, et al. Bioorg Med Chem. 2011 Jan 15;19(2):771-82. doi: 10.1016/j.bmc.2010.12.023. Epub 2010 Dec 13. Bioorg Med Chem. 2011. PMID: 21215640

7

Modulation of PPAR receptor subtype selectivity of the ligands: aliphatic chain vs aromatic ring as a spacer between pharmacophore and the lipophilic moiety.

Pingali H, Jain M, Shah S, Patil P, Makadia P, Zaware P, Sairam KV, Jamili J, Goel A, Patel M, Patel P. Pingali H, et al. Among authors: makadia p. Bioorg Med Chem Lett. 2008 Dec 15;18(24):6471-5. doi: 10.1016/j.bmcl.2008.10.062. Epub 2008 Oct 17. Bioorg Med Chem Lett. 2008. PMID: 18976908

8

Novel oxazole containing phenylpropane derivatives as peroxisome proliferator activated receptor agonists with hypolipidemic activity.

Pingali H, Raval S, Raval P, Makadia P, Zaware P, Goel A, Suthar D, Jain M, Patel P. Pingali H, et al. Among authors: makadia p. Pharmazie. 2008 Jul;63(7):497-502. Pharmazie. 2008. PMID: 18717481

9

Peroperative Intra-Articular Infiltration of Tranexamic Acid and Ropivacaine Cocktail in Patients Undergoing Total Knee Arthroplasty: A Randomized Controlled Trial.

Singh H, Agarwal KK, Tyagi S, Makadia P, Oza B, Jain P, Patel M. Singh H, et al. Among authors: makadia p. Cureus. 2022 Mar 12;14(3):e23091. doi: 10.7759/cureus.23091. eCollection 2022 Mar. Cureus. 2022. PMID: 35464570 Free PMC article.

10

Optogenetic Activation of Colon Epithelium of the Mouse Produces High-Frequency Bursting in Extrinsic Colon Afferents and Engages Visceromotor Responses.

Makadia PA, Najjar SA, Saloman JL, Adelman P, Feng B, Margiotta JF, Albers KM, Davis BM. Makadia PA, et al. J Neurosci. 2018 Jun 20;38(25):5788-5798. doi: 10.1523/JNEUROSCI.0837-18.2018. Epub 2018 May 22. J Neurosci. 2018. PMID: 29789376 Free PMC article.

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