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Discovery of isoxazolyl-based inhibitors of Plasmodium falciparum cGMP-dependent protein kinase.
RSC Med Chem. 2019 Dec 16;11(1):98-101. doi: 10.1039/c9md00511k. eCollection 2020 Jan 1.
RSC Med Chem. 2019.
PMID: 33479608
Free PMC article.
Discovery of a Stress-Activated Protein Kinase Inhibitor for Lymphatic Filariasis.
Tummalapalli SR, Bhat R, Chojnowski A, Prorok M, Kreiss T, Goldberg R, Canan S, Hawryluk N, Mortensen D, Khetani V, Zeldis J, Siekierka JJ, Rotella DP.
Tummalapalli SR, et al. Among authors: kreiss t.
ACS Med Chem Lett. 2018 Feb 9;9(3):210-214. doi: 10.1021/acsmedchemlett.7b00477. eCollection 2018 Mar 8.
ACS Med Chem Lett. 2018.
PMID: 29541362
Free PMC article.
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Discovery of Imidazole-Based Inhibitors of Plasmodium falciparum cGMP-Dependent Protein Kinase.
Bheemanaboina RRY, de Souza ML, Gonzalez ML, Mahmood SU, Eck T, Kreiss T, Aylor SO, Roth A, Lee P, Pybus BS, Colussi DJ, Childers WE, Gordon J, Siekierka JJ, Bhanot P, Rotella DP.
Bheemanaboina RRY, et al. Among authors: kreiss t.
ACS Med Chem Lett. 2021 Nov 15;12(12):1962-1967. doi: 10.1021/acsmedchemlett.1c00540. eCollection 2021 Dec 9.
ACS Med Chem Lett. 2021.
PMID: 34917261
Free PMC article.
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Characterization of Competitive Inhibitors of Plasmodium falciparum cGMP-Dependent Protein Kinase.
Eck T, Laureano de Souza M, Delvillar M, Ashraf K, Yadav Bheemanaboina RR, Chakrasali R, Kreiss T, Siekierka JJ, Rotella DP, Bhanot P, Goodey NM.
Eck T, et al. Among authors: kreiss t.
Chembiochem. 2022 Apr 5;23(7):e202100704. doi: 10.1002/cbic.202100704. Epub 2022 Feb 23.
Chembiochem. 2022.
PMID: 35044710
Free PMC article.
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A novel series of putative Brugia malayi histone demethylase inhibitors as potential anti-filarial drugs.
Kreiss T, Eck T, Hart B, Tummalapalli S, Rotella D, Siekierka J.
Kreiss T, et al.
PLoS Negl Trop Dis. 2022 Mar 16;16(3):e0010216. doi: 10.1371/journal.pntd.0010216. eCollection 2022 Mar.
PLoS Negl Trop Dis. 2022.
PMID: 35294431
Free PMC article.
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Filarial nematode phenotypic screening cascade to identify compounds with anti-parasitic activity for drug discovery optimization.
Hawryluk N, Zhiru L, Carlow C, Gokool S, Townson S, Kreiss T, Chojnowski A, Prorok M, Siekierka J, Ehrens A, Koschel M, Lhermitte-Vallarino N, Martin C, Hoerauf A, Hernandez G, Canan S, Khetani V, Zeldis J, Specht S, Hübner MP, Scandale I.
Hawryluk N, et al. Among authors: kreiss t.
Int J Parasitol Drugs Drug Resist. 2022 Aug;19:89-97. doi: 10.1016/j.ijpddr.2022.06.002. Epub 2022 Jun 23.
Int J Parasitol Drugs Drug Resist. 2022.
PMID: 35834918
Free PMC article.
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Phosphatidylserine-Targeting Monoclonal Antibodies Exhibit Distinct Biochemical and Cellular Effects on Anti-CD3/CD28-Stimulated T Cell IFN-γ and TNF-α Production.
Calianese D, Kreiss T, Kasikara C, Davra V, Lahey KC, Gadiyar V, Geng K, Singh S, Honnen W, Jaijyan DK, Reichman C, Siekierka J, Gennaro ML, Kotenko SV, Ucker DS, Brekken RA, Pinter A, Birge RB, Choudhary A.
Calianese D, et al. Among authors: kreiss t.
J Immunol. 2021 Jul 15;207(2):436-448. doi: 10.4049/jimmunol.2000763. Epub 2021 Jul 2.
J Immunol. 2021.
PMID: 34215655
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