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HER2 Kinase-Targeted Breast Cancer Therapy: Design, Synthesis, and In Vitro and In Vivo Evaluation of Novel Lapatinib Congeners as Selective and Potent HER2 Inhibitors with Favorable Metabolic Stability.
J Med Chem. 2020 Dec 24;63(24):15906-15945. doi: 10.1021/acs.jmedchem.0c01647. Epub 2020 Dec 14.
J Med Chem. 2020.
PMID: 33314925
4-Substituted-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine derivatives: design, synthesis, antitumor and EGFR tyrosine kinase inhibitory activity.
Abbas SE, Aly EI, Awadallah FM, Mahmoud WR.
Abbas SE, et al. Among authors: aly ei.
Chem Biol Drug Des. 2015 May;85(5):608-22. doi: 10.1111/cbdd.12451. Epub 2014 Nov 14.
Chem Biol Drug Des. 2015.
PMID: 25318985
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Synthesis and biological activity of 2,5-diaryl-3-methylpyrimido[4,5-c]quinolin-1(2H)-one derivatives.
Metwally K, Aly O, Aly E, Banerjee A, Ravindra R, Bane S.
Metwally K, et al.
Bioorg Med Chem. 2007 Mar 15;15(6):2434-40. doi: 10.1016/j.bmc.2007.01.016. Epub 2007 Jan 17.
Bioorg Med Chem. 2007.
PMID: 17275318
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Corrigendum to "Synthesis and biological activity of 2,5-diaryl-3-methylpyrimido[4,5-c]quinolin-1(2H)-one derivatives" [Bioorg. Med. Chem. 15 (2007) 2434-2440].
Metwally K, Aly O, Aly E, Banerjee A, Ravindra R, Bane S.
Metwally K, et al.
Bioorg Med Chem. 2017 May 1;25(9):2679. doi: 10.1016/j.bmc.2017.03.025. Epub 2017 Mar 22.
Bioorg Med Chem. 2017.
PMID: 28341404
No abstract available.
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Synthesis and antitubercular activity of 6-chloro (unsubstituted)- 2-methoxy-9-substituted acridine derivatives.
Aly EI, Abadi AH.
Aly EI, et al.
Arch Pharm Res. 2004 Jul;27(7):713-9. doi: 10.1007/BF02980137.
Arch Pharm Res. 2004.
PMID: 15356996
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