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New Small-Molecule Glycoconjugates of Docetaxel and GalNAc for Targeted Delivery to Hepatocellular Carcinoma.
Petrov RA, Mefedova SR, Yamansarov EY, Maklakova SY, Grishin DA, Lopatukhina EV, Burenina OY, Lopukhov AV, Kovalev SV, Timchenko YV, Ondar EE, Ivanenkov YA, Evteev SA, Vaneev AN, Timoshenko RV, Klyachko NL, Erofeev AS, Gorelkin PV, Beloglazkina EK, Majouga AG. Petrov RA, et al. Among authors: lopukhov av. Mol Pharm. 2021 Jan 4;18(1):461-468. doi: 10.1021/acs.molpharmaceut.0c00980. Epub 2020 Dec 2. Mol Pharm. 2021. PMID: 33264010
Synthesis and Evaluation of New Trivalent Ligands for Hepatocyte Targeting via the Asialoglycoprotein Receptor.
Reshitko GS, Yamansarov EY, Evteev SA, Lopatukhina EV, Shkil' DO, Saltykova IV, Lopukhov AV, Kovalev SV, Lobov AN, Kislyakov IV, Burenina OY, Klyachko NL, Garanina AS, Dontsova OA, Ivanenkov YA, Erofeev AS, Gorelkin PV, Beloglazkina EK, Majouga AG. Reshitko GS, et al. Among authors: lopukhov av. Bioconjug Chem. 2020 May 20;31(5):1313-1319. doi: 10.1021/acs.bioconjchem.0c00202. Epub 2020 May 9. Bioconjug Chem. 2020. PMID: 32379426
Mannosylated Cationic Copolymers for Gene Delivery to Macrophages.
Lopukhov AV, Yang Z, Haney MJ, Bronich TK, Sokolsky-Papkov M, Batrakova EV, Klyachko NL, Kabanov AV. Lopukhov AV, et al. Macromol Biosci. 2021 Apr;21(4):e2000371. doi: 10.1002/mabi.202000371. Epub 2021 Feb 22. Macromol Biosci. 2021. PMID: 33615675 Free PMC article.
Discovery of Bivalent GalNAc-Conjugated Betulin as a Potent ASGPR-Directed Agent against Hepatocellular Carcinoma.
Yamansarov EY, Lopatukhina EV, Evteev SA, Skvortsov DA, Lopukhov AV, Kovalev SV, Vaneev AN, Shkil' DO, Akasov RA, Lobov AN, Naumenko VA, Pavlova EN, Ryabaya OO, Burenina OY, Ivanenkov YA, Klyachko NL, Erofeev AS, Gorelkin PV, Beloglazkina EK, Majouga AG. Yamansarov EY, et al. Among authors: lopukhov av. Bioconjug Chem. 2021 Apr 21;32(4):763-781. doi: 10.1021/acs.bioconjchem.1c00042. Epub 2021 Mar 10. Bioconjug Chem. 2021. PMID: 33691403
Novel His-tag Variants for Insertion Inside Polypeptide Chain.
Tarabarova AG, Lopukhov A, Fedorov AN, Yurkova MS. Tarabarova AG, et al. ACS Omega. 2023 Dec 22;9(1):858-865. doi: 10.1021/acsomega.3c06682. eCollection 2024 Jan 9. ACS Omega. 2023. PMID: 38222536 Free PMC article.
Production of a Cloned Offspring and CRISPR/Cas9 Genome Editing of Embryonic Fibroblasts in Cattle.
Singina GN, Sergiev PV, Lopukhov AV, Rubtsova MP, Taradajnic NP, Ravin NV, Shedova EN, Taradajnic TE, Polejaeva IA, Dozev AV, Brem G, Dontsova OA, Zinovieva NA. Singina GN, et al. Among authors: lopukhov av. Dokl Biochem Biophys. 2021 May;496(1):48-51. doi: 10.1134/S1607672921010099. Epub 2021 Mar 10. Dokl Biochem Biophys. 2021. PMID: 33689075 Free PMC article.
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