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Identification of a Potent and Selective 5-HT1A Receptor Agonist with In Vitro and In Vivo Antinociceptive Activity.
Linciano P, Sorbi C, Comitato A, Lesniak A, Bujalska-Zadrożny M, Pawłowska A, Bielenica A, Orzelska-Górka J, Kędzierska E, Biała G, Ronsisvalle S, Limoncella S, Casarini L, Cichero E, Fossa P, Satała G, Bojarski AJ, Brasili L, Bardoni R, Franchini S. Linciano P, et al. Among authors: kedzierska e. ACS Chem Neurosci. 2020 Dec 16;11(24):4111-4127. doi: 10.1021/acschemneuro.0c00289. Epub 2020 Dec 2. ACS Chem Neurosci. 2020. PMID: 33263393 Free PMC article.
Synthesis, in vitro and in vivo pharmacological evaluation of serotoninergic ligands containing an isonicotinic nucleus.
Fiorino F, Ciano A, Magli E, Severino B, Corvino A, Perissutti E, Frecentese F, Di Vaio P, Izzo AA, Capasso R, Massarelli P, Nencini C, Rossi I, Kędzierska E, Orzelska-Gòrka J, Bielenica A, Santagada V, Caliendo G. Fiorino F, et al. Among authors: kedzierska e. Eur J Med Chem. 2016 Mar 3;110:133-50. doi: 10.1016/j.ejmech.2016.01.021. Epub 2016 Jan 18. Eur J Med Chem. 2016. PMID: 26820556
5-HT2 receptor affinity, docking studies and pharmacological evaluation of a series of 1,3-disubstituted thiourea derivatives.
Bielenica A, Kędzierska E, Koliński M, Kmiecik S, Koliński A, Fiorino F, Severino B, Magli E, Corvino A, Rossi I, Massarelli P, Kozioł AE, Sawczenko A, Struga M. Bielenica A, et al. Among authors: kedzierska e. Eur J Med Chem. 2016 Jun 30;116:173-186. doi: 10.1016/j.ejmech.2016.03.073. Epub 2016 Mar 30. Eur J Med Chem. 2016. PMID: 27061981
In Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048).
Aaltonen N, Kedzierska E, Orzelska-Górka J, Lehtonen M, Navia-Paldanius D, Jakupovic H, Savinainen JR, Nevalainen T, Laitinen JT, Parkkari T, Gynther M. Aaltonen N, et al. Among authors: kedzierska e. J Pharmacol Exp Ther. 2016 Oct;359(1):62-72. doi: 10.1124/jpet.116.233114. Epub 2016 Jul 22. J Pharmacol Exp Ther. 2016. PMID: 27451409
New 5-HT1A, 5HT2A and 5HT2C receptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation.
Fiorino F, Magli E, Kędzierska E, Ciano A, Corvino A, Severino B, Perissutti E, Frecentese F, Di Vaio P, Saccone I, Izzo AA, Capasso R, Massarelli P, Rossi I, Orzelska-Gòrka J, Kotlińska JH, Santagada V, Caliendo G. Fiorino F, et al. Among authors: kedzierska e. Bioorg Med Chem. 2017 Oct 15;25(20):5820-5837. doi: 10.1016/j.bmc.2017.09.018. Epub 2017 Sep 18. Bioorg Med Chem. 2017. PMID: 28943244
66 results