Pockes S - Search Results

1

A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.

Höring C, Seibel U, Tropmann K, Grätz L, Mönnich D, Pitzl S, Bernhardt G, Pockes S, Strasser A. Höring C, et al. Among authors: pockes s. Int J Mol Sci. 2020 Nov 10;21(22):8440. doi: 10.3390/ijms21228440. Int J Mol Sci. 2020. PMID: 33182741 Free PMC article.

2

Synthesis, biological evaluation, and computational studies of Tri- and tetracyclic nitrogen-bridgehead compounds as potent dual-acting AChE inhibitors and hH3 receptor antagonists.

Darras FH, Pockes S, Huang G, Wehle S, Strasser A, Wittmann HJ, Nimczick M, Sotriffer CA, Decker M. Darras FH, et al. Among authors: pockes s. ACS Chem Neurosci. 2014 Mar 19;5(3):225-42. doi: 10.1021/cn4002126. Epub 2014 Jan 14. ACS Chem Neurosci. 2014. PMID: 24422467 Free PMC article.

3

Development of a Conformational Histamine H₃ Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists.

Schihada H, Ma X, Zabel U, Vischer HF, Schulte G, Leurs R, Pockes S, Lohse MJ. Schihada H, et al. Among authors: pockes s. ACS Sens. 2020 Jun 26;5(6):1734-1742. doi: 10.1021/acssensors.0c00397. Epub 2020 May 28. ACS Sens. 2020. PMID: 32397705 Free PMC article.

4

NanoBRET binding assay for histamine H₂ receptor ligands using live recombinant HEK293T cells.

Grätz L, Tropmann K, Bresinsky M, Müller C, Bernhardt G, Pockes S. Grätz L, et al. Among authors: pockes s. Sci Rep. 2020 Aug 6;10(1):13288. doi: 10.1038/s41598-020-70332-3. Sci Rep. 2020. PMID: 32764682 Free PMC article.

5

A Split Luciferase Complementation Assay for the Quantification of β-Arrestin2 Recruitment to Dopamine D₂-Like Receptors.

Forster L, Grätz L, Mönnich D, Bernhardt G, Pockes S. Forster L, et al. Among authors: pockes s. Int J Mol Sci. 2020 Aug 24;21(17):6103. doi: 10.3390/ijms21176103. Int J Mol Sci. 2020. PMID: 32847148 Free PMC article.

6

Discovery of a G Protein-Biased Radioligand for the Histamine H₂ Receptor with Reversible Binding Properties.

Tropmann K, Höring C, Plank N, Pockes S. Tropmann K, et al. Among authors: pockes s. J Med Chem. 2020 Nov 12;63(21):13090-13102. doi: 10.1021/acs.jmedchem.0c01494. Epub 2020 Oct 27. J Med Chem. 2020. PMID: 33108724

7

Structural modifications in the distal, regulatory region of histamine H₃ receptor antagonists leading to the identification of a potent anti-obesity agent.

Szczepańska K, Pockes S, Podlewska S, Höring C, Mika K, Latacz G, Bednarski M, Siwek A, Karcz T, Nagl M, Bresinsky M, Mönnich D, Seibel U, Kuder KJ, Kotańska M, Stark H, Elz S, Kieć-Kononowicz K. Szczepańska K, et al. Among authors: pockes s. Eur J Med Chem. 2021 Mar 5;213:113041. doi: 10.1016/j.ejmech.2020.113041. Epub 2020 Nov 24. Eur J Med Chem. 2021. PMID: 33261900

8

Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H₂R and D₃R.

Biselli S, Bresinsky M, Tropmann K, Forster L, Honisch C, Buschauer A, Bernhardt G, Pockes S. Biselli S, et al. Among authors: pockes s. Eur J Med Chem. 2021 Mar 15;214:113190. doi: 10.1016/j.ejmech.2021.113190. Epub 2021 Jan 19. Eur J Med Chem. 2021. PMID: 33548637

9

Histamine H₂ receptor radioligands: triumphs and challenges.

Pockes S, Tropmann K. Pockes S, et al. Future Med Chem. 2021 Jun;13(12):1073-1081. doi: 10.4155/fmc-2021-0058. Epub 2021 Apr 28. Future Med Chem. 2021. PMID: 33906421 Free article. Review.

10

Author Correction: NanoBRET binding assay for histamine H₂ receptor ligands using live recombinant HEK293T cells.

Grätz L, Tropmann K, Bresinsky M, Müller C, Bernhardt G, Pockes S. Grätz L, et al. Among authors: pockes s. Sci Rep. 2021 May 18;11(1):10747. doi: 10.1038/s41598-021-89954-2. Sci Rep. 2021. PMID: 34006951 Free PMC article. No abstract available.

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