Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
6 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Discovery of New Heterocyclic Ring Systems as Novel and Potent V1A Receptor Antagonists.
ACS Chem Neurosci. 2020 Nov 4;11(21):3532-3540. doi: 10.1021/acschemneuro.0c00486. Epub 2020 Oct 21.
ACS Chem Neurosci. 2020.
PMID: 33084311
New V1a receptor antagonist. Part 2. Identification and optimization of triazolobenzazepines.
Bozó É, Baska F, Lövei K, Szántó G, Domány-Kovács K, Kurkó D, Szondiné Kordás K, Szokoli T, Bata I.
Bozó É, et al. Among authors: domany kovacs k.
Bioorg Med Chem Lett. 2020 Sep 15;30(18):127417. doi: 10.1016/j.bmcl.2020.127417. Epub 2020 Jul 21.
Bioorg Med Chem Lett. 2020.
PMID: 32731087
Item in Clipboard
New V1a receptor antagonist. Part 1. Synthesis and SAR development of urea derivatives.
Szántó G, Makó A, Baska F, Bozó É, Domány-Kovács K, Kurkó D, Cselenyák A, Mohácsi R, Kordás KS, Bata I.
Szántó G, et al. Among authors: domany kovacs k.
Bioorg Med Chem Lett. 2020 Sep 15;30(18):127416. doi: 10.1016/j.bmcl.2020.127416. Epub 2020 Jul 24.
Bioorg Med Chem Lett. 2020.
PMID: 32736211
Item in Clipboard
Synthesis and Characterization of New V1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers.
Szeleczky Z, Szakács Z, Bozó É, Baska F, Vukics K, Lévai S, Temesvári K, Vass E, Béni Z, Krámos B, Magdó I, Szántay C Jr, Kóti J, Domány-Kovács K, Greiner I, Bata I.
Szeleczky Z, et al. Among authors: domany kovacs k.
J Med Chem. 2021 Jul 22;64(14):10445-10468. doi: 10.1021/acs.jmedchem.1c00863. Epub 2021 Jul 13.
J Med Chem. 2021.
PMID: 34255509
Item in Clipboard
Controlling receptor function from the extracellular vestibule of G-protein coupled receptors.
Egyed A , Domány-Kovács K , Koványi B , Horti F , Kurkó D , Kiss DJ , Pándy-Szekeres G , Greiner I , Keserű GM .
Egyed A , et al. Among authors: domany kovacs k.
Chem Commun (Camb). 2020 Nov 25;56(91):14167-14170. doi: 10.1039/d0cc05532h. Epub 2020 Oct 20.
Chem Commun (Camb). 2020.
PMID: 33079104
Item in Clipboard
Discovery and Characterization of RGH-122, a Potent, Selective, and Orally Bioavailable V1a Receptor Antagonist.
Baska F, Bozó É, Szeleczky Z, Szántó G, Vukics K, Szakács Z, Domány-Kovács K, Kurkó D, Vass E, Thán M, Vastag M, Temesvári K, Lévai S, Halász AS, Szondiné Kordás K, Román V, Greiner I, Bata I.
Baska F, et al. Among authors: domany kovacs k.
J Med Chem. 2024 Jan 11;67(1):643-673. doi: 10.1021/acs.jmedchem.3c01868. Epub 2024 Jan 2.
J Med Chem. 2024.
PMID: 38165765
Item in Clipboard
Cite
Cite