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Page 1
Discovery of New Heterocyclic Ring Systems as Novel and Potent V1A Receptor Antagonists.
Baska F, Szántó G, Bozó É, Szakács Z, Dékány M, Szondiné Kordás K, Domány-Kovács K, Kurkó D, Hodoscsek B, Magdó I, Krámos B, Béni Z, Vastag M, Bata I. Baska F, et al. Among authors: bozo e. ACS Chem Neurosci. 2020 Nov 4;11(21):3532-3540. doi: 10.1021/acschemneuro.0c00486. Epub 2020 Oct 21. ACS Chem Neurosci. 2020. PMID: 33084311
Selective NR1/2B N-methyl-D-aspartate receptor antagonists among indole-2-carboxamides and benzimidazole-2-carboxamides.
Borza I, Bozó E, Barta-Szalai G, Kiss C, Tárkányi G, Demeter A, Gáti T, Háda V, Kolok S, Gere A, Fodor L, Nagy J, Galgóczy K, Magdó I, Agai B, Fetter J, Bertha F, Keserü GM, Horváth C, Farkas S, Greiner I, Domány G. Borza I, et al. Among authors: bozo e. J Med Chem. 2007 Mar 8;50(5):901-14. doi: 10.1021/jm060420k. Epub 2007 Feb 10. J Med Chem. 2007. PMID: 17290978
Quinolinyl- and phenantridinyl-acetamides as bradykinin B1 receptor antagonists.
Eles J, Beke G, Vágó I, Bozó E, Huszár J, Tarcsay A, Kolok S, Schmidt E, Vastag M, Hornok K, Farkas S, Domány G, Keserű GM. Eles J, et al. Among authors: bozo e. Bioorg Med Chem Lett. 2012 May 1;22(9):3095-9. doi: 10.1016/j.bmcl.2012.03.065. Epub 2012 Mar 21. Bioorg Med Chem Lett. 2012. PMID: 22483585
Discovery of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor: Scaffold hopping approach.
Ledneczki I, Tapolcsányi P, Gábor E, Visegrády A, Vass M, Éles J, Holm P, Horváth A, Pocsai A, Mahó S, Greiner I, Krámos B, Béni Z, Kóti J, Káncz AE, Thán M, Kolok S, Laszy J, Balázs O, Bugovits G, Nagy J, Vastag M, Szájli Á, Bozó É, Lévay G, Lendvai B, Némethy Z. Ledneczki I, et al. Among authors: bozo e. Eur J Med Chem. 2021 Mar 15;214:113189. doi: 10.1016/j.ejmech.2021.113189. Epub 2021 Jan 14. Eur J Med Chem. 2021. PMID: 33540354
Synthesis and Characterization of New V1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers.
Szeleczky Z, Szakács Z, Bozó É, Baska F, Vukics K, Lévai S, Temesvári K, Vass E, Béni Z, Krámos B, Magdó I, Szántay C Jr, Kóti J, Domány-Kovács K, Greiner I, Bata I. Szeleczky Z, et al. Among authors: bozo e. J Med Chem. 2021 Jul 22;64(14):10445-10468. doi: 10.1021/acs.jmedchem.1c00863. Epub 2021 Jul 13. J Med Chem. 2021. PMID: 34255509
Vasopressin receptor antagonists: a patent summary (2018-2022).
Baska F, Bozó É, Patócs T. Baska F, et al. Among authors: bozo e. Expert Opin Ther Pat. 2023 Jan-Jun;33(5):385-395. doi: 10.1080/13543776.2023.2218546. Epub 2023 May 29. Expert Opin Ther Pat. 2023. PMID: 37226495 Review.
Discovery and Characterization of RGH-122, a Potent, Selective, and Orally Bioavailable V1a Receptor Antagonist.
Baska F, Bozó É, Szeleczky Z, Szántó G, Vukics K, Szakács Z, Domány-Kovács K, Kurkó D, Vass E, Thán M, Vastag M, Temesvári K, Lévai S, Halász AS, Szondiné Kordás K, Román V, Greiner I, Bata I. Baska F, et al. Among authors: bozo e. J Med Chem. 2024 Jan 11;67(1):643-673. doi: 10.1021/acs.jmedchem.3c01868. Epub 2024 Jan 2. J Med Chem. 2024. PMID: 38165765
Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists.
Borza I, Kolok S, Gere A, Agai-Csongor E, Agai B, Tárkányi G, Horváth C, Barta-Szalai G, Bozó E, Kiss C, Bielik A, Nagy J, Farkas S, Domány G. Borza I, et al. Among authors: bozo e. Bioorg Med Chem Lett. 2003 Nov 3;13(21):3859-61. doi: 10.1016/s0960-894x(03)00708-x. Bioorg Med Chem Lett. 2003. PMID: 14552795
31 results