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Protein kinase inhibitors for amyotrophic lateral sclerosis therapy.
Br J Pharmacol. 2021 Mar;178(6):1316-1335. doi: 10.1111/bph.15221. Epub 2020 Aug 31.
Br J Pharmacol. 2021.
PMID: 32737989
Free article.
Review.
Therapeutic potential of novel Cell Division Cycle Kinase 7 inhibitors on TDP-43-related pathogenesis such as Frontotemporal Lobar Degeneration (FTLD) and amyotrophic lateral sclerosis (ALS).
Vaca G, Martinez-Gonzalez L, Fernandez A, Rojas-Prats E, Porras G, Cuevas EP, Gil C, Martinez A, Martin-Requero Á.
Vaca G, et al. Among authors: rojas prats e.
J Neurochem. 2021 Feb;156(3):379-390. doi: 10.1111/jnc.15118. Epub 2020 Jul 17.
J Neurochem. 2021.
PMID: 32628315
Free article.
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Targeting nuclear protein TDP-43 by cell division cycle kinase 7 inhibitors: A new therapeutic approach for amyotrophic lateral sclerosis.
Rojas-Prats E, Martinez-Gonzalez L, Gonzalo-Consuegra C, Liachko NF, Perez C, Ramírez D, Kraemer BC, Martin-Requero Á, Perez DI, Gil C, de Lago E, Martinez A.
Rojas-Prats E, et al.
Eur J Med Chem. 2021 Jan 15;210:112968. doi: 10.1016/j.ejmech.2020.112968. Epub 2020 Oct 28.
Eur J Med Chem. 2021.
PMID: 33139113
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Druggable cavities and allosteric modulators of the cell division cycle 7 (CDC7) kinase.
Rojas-Prats E, Martinez-Gonzalez L, Gil C, Ramírez D, Martinez A.
Rojas-Prats E, et al.
J Enzyme Inhib Med Chem. 2024 Dec;39(1):2301767. doi: 10.1080/14756366.2024.2301767. Epub 2024 Jan 11.
J Enzyme Inhib Med Chem. 2024.
PMID: 38205514
Free PMC article.
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Improved Controlled Release and Brain Penetration of the Small Molecule S14 Using PLGA Nanoparticles.
Nozal V, Rojas-Prats E, Maestro I, Gil C, Perez DI, Martinez A.
Nozal V, et al. Among authors: rojas prats e.
Int J Mol Sci. 2021 Mar 22;22(6):3206. doi: 10.3390/ijms22063206.
Int J Mol Sci. 2021.
PMID: 33809846
Free PMC article.
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Increasing Brain Permeability of PHA-767491, a Cell Division Cycle 7 Kinase Inhibitor, with Biodegradable Polymeric Nanoparticles.
Rojas-Prats E, Tosat-Bitrián C, Martínez-González L, Nozal V, Pérez DI, Martínez A.
Rojas-Prats E, et al.
Pharmaceutics. 2021 Jan 28;13(2):180. doi: 10.3390/pharmaceutics13020180.
Pharmaceutics. 2021.
PMID: 33525757
Free PMC article.
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