Kieffer C - Search Results

1

Noncellular screening for the discovery of protein-protein interaction modulators.

Kieffer C, Jourdan JP, Jouanne M, Voisin-Chiret AS. Kieffer C, et al. Drug Discov Today. 2020 Sep;25(9):1592-1603. doi: 10.1016/j.drudis.2020.07.012. Epub 2020 Jul 16. Drug Discov Today. 2020. PMID: 32682931 Review.

2

PROTAC technology: A new drug design for chemical biology with many challenges in drug discovery.

Guedeney N, Cornu M, Schwalen F, Kieffer C, Voisin-Chiret AS. Guedeney N, et al. Among authors: kieffer c. Drug Discov Today. 2023 Jan;28(1):103395. doi: 10.1016/j.drudis.2022.103395. Epub 2022 Oct 10. Drug Discov Today. 2023. PMID: 36228895 Review.

3

Computational Tool to Design Small Synthetic Inhibitors Selective for XIAP-BIR3 Domain.

Farag M, Kieffer C, Guedeney N, Voisin-Chiret AS, Sopkova-de Oliveira Santos J. Farag M, et al. Among authors: kieffer c. Molecules. 2023 Jun 30;28(13):5155. doi: 10.3390/molecules28135155. Molecules. 2023. PMID: 37446817 Free PMC article.

4

Molecular glue degraders: exciting opportunities for novel drug discovery.

Lemaitre T, Cornu M, Schwalen F, Since M, Kieffer C, Voisin-Chiret AS. Lemaitre T, et al. Among authors: kieffer c. Expert Opin Drug Discov. 2024 Apr;19(4):433-449. doi: 10.1080/17460441.2024.2306845. Epub 2024 Jan 24. Expert Opin Drug Discov. 2024. PMID: 38240114 Review.

5

Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents.

Primas N, Suzanne P, Verhaeghe P, Hutter S, Kieffer C, Laget M, Cohen A, Broggi J, Lancelot JC, Lesnard A, Dallemagne P, Rathelot P, Rault S, Vanelle P, Azas N. Primas N, et al. Among authors: kieffer c. Eur J Med Chem. 2014 Aug 18;83:26-35. doi: 10.1016/j.ejmech.2014.06.014. Epub 2014 Jun 10. Eur J Med Chem. 2014. PMID: 24946216

6

A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: a structure-activity relationship study of antiplasmodial activity.

Primas N, Verhaeghe P, Cohen A, Kieffer C, Dumètre A, Hutter S, Rault S, Rathelot P, Azas N, Vanelle P. Primas N, et al. Among authors: kieffer c. Molecules. 2012 Jul 5;17(7):8105-17. doi: 10.3390/molecules17078105. Molecules. 2012. PMID: 22766802 Free PMC article.

7

Preventing the contamination of hospital personnel by cytotoxic agents: evaluation and training of the para-professional healthcare workers in oncology units.

Kieffer C, Verhaeghe P, Lagrassa S, Grégoire R, Moussaoui Z, Casteras-Ducros C, Clark JE, Vanelle P, Rathelot P. Kieffer C, et al. Eur J Cancer Care (Engl). 2015 May;24(3):404-10. doi: 10.1111/ecc.12249. Epub 2014 Oct 7. Eur J Cancer Care (Engl). 2015. PMID: 25289934

8

Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold.

Desroches J, Kieffer C, Primas N, Hutter S, Gellis A, El-Kashef H, Rathelot P, Verhaeghe P, Azas N, Vanelle P. Desroches J, et al. Among authors: kieffer c. Eur J Med Chem. 2017 Jan 5;125:68-86. doi: 10.1016/j.ejmech.2016.09.029. Epub 2016 Sep 10. Eur J Med Chem. 2017. PMID: 27654395

9

Target fishing reveals PfPYK-1 and PfRab6 as potential targets of an antiplasmodial 4-anilino-2-trichloromethylquinazoline hit compound.

Kieffer C, Primas N, Hutter S, Merckx A, Reininger L, Bach S, Ruchaud S, Gaillard F, Laget M, Amrane D, Hervé L, Castera-Ducros C, Renault J, Dumètre A, Rault S, Doerig C, Rathelot P, Vanelle P, Azas N, Verhaeghe P. Kieffer C, et al. Bioorg Med Chem. 2024 Mar 15;102:117654. doi: 10.1016/j.bmc.2024.117654. Epub 2024 Feb 28. Bioorg Med Chem. 2024. PMID: 38452406

10

Looking for new antileishmanial derivatives in 8-nitroquinolin-2(1H)-one series.

Kieffer C, Cohen A, Verhaeghe P, Hutter S, Castera-Ducros C, Laget M, Remusat V, M'Rabet MK, Rault S, Rathelot P, Azas N, Vanelle P. Kieffer C, et al. Eur J Med Chem. 2015 Mar 6;92:282-94. doi: 10.1016/j.ejmech.2014.12.056. Epub 2014 Dec 31. Eur J Med Chem. 2015. PMID: 25559208

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