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Multiparameter Kinetic Analysis for Covalent Fragment Optimization by Using Quantitative Irreversible Tethering (qIT).
Chembiochem. 2020 Dec 1;21(23):3417-3422. doi: 10.1002/cbic.202000457. Epub 2020 Aug 7.
Chembiochem. 2020.
PMID: 32659037
Free PMC article.
How can the potential of the duocarmycins be unlocked for cancer therapy?
Jukes Z, Morais GR, Loadman PM, Pors K.
Jukes Z, et al.
Drug Discov Today. 2021 Feb;26(2):577-584. doi: 10.1016/j.drudis.2020.11.020. Epub 2020 Nov 21.
Drug Discov Today. 2021.
PMID: 33232841
Review.
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