Trapencieris P - Search Results

1

Bicyclic Boronates as Potent Inhibitors of AmpC, the Class C β-Lactamase from Escherichia coli.

Lang PA, Parkova A, Leissing TM, Calvopiña K, Cain R, Krajnc A, Panduwawala TD, Philippe J, Fishwick CWG, Trapencieris P, Page MGP, Schofield CJ, Brem J. Lang PA, et al. Among authors: trapencieris p. Biomolecules. 2020 Jun 12;10(6):899. doi: 10.3390/biom10060899. Biomolecules. 2020. PMID: 32545682 Free PMC article.

2

Broad Spectrum β-Lactamase Inhibition by a Thioether Substituted Bicyclic Boronate.

Parkova A, Lucic A, Krajnc A, Brem J, Calvopiña K, Langley GW, McDonough MA, Trapencieris P, Schofield CJ. Parkova A, et al. Among authors: trapencieris p. ACS Infect Dis. 2020 Jun 12;6(6):1398-1404. doi: 10.1021/acsinfecdis.9b00330. Epub 2020 Jan 6. ACS Infect Dis. 2020. PMID: 31841636

3

Structures of plasmepsin II from Plasmodium falciparum in complex with two hydroxyethylamine-based inhibitors.

Recacha R, Leitans J, Akopjana I, Aprupe L, Trapencieris P, Jaudzems K, Jirgensons A, Tars K. Recacha R, et al. Among authors: trapencieris p. Acta Crystallogr F Struct Biol Commun. 2015 Dec;71(Pt 12):1531-9. doi: 10.1107/S2053230X15022049. Epub 2015 Nov 27. Acta Crystallogr F Struct Biol Commun. 2015. PMID: 26625296 Free PMC article.

4

5-membered cyclic hydroxamic acids as HDAC inhibitors.

Mutule I, Borovika D, Rozenberga E, Romanchikova N, Zalubovskis R, Shestakova I, Trapencieris P. Mutule I, et al. Among authors: trapencieris p. J Enzyme Inhib Med Chem. 2015 Apr;30(2):216-23. doi: 10.3109/14756366.2014.912214. Epub 2014 Jun 18. J Enzyme Inhib Med Chem. 2015. PMID: 24939099

5

Pyrazole-based inhibitors of enhancer of zeste homologue 2 induce apoptosis and autophagy in cancer cells.

Mellini P, Marrocco B, Borovika D, Polletta L, Carnevale I, Saladini S, Stazi G, Zwergel C, Trapencieris P, Ferretti E, Tafani M, Valente S, Mai A. Mellini P, et al. Among authors: trapencieris p. Philos Trans R Soc Lond B Biol Sci. 2018 Jun 5;373(1748):20170150. doi: 10.1098/rstb.2017.0150. Philos Trans R Soc Lond B Biol Sci. 2018. PMID: 29685965 Free PMC article.

6

Saccharin sulfonamides as inhibitors of carbonic anhydrases I, II, VII, XII, and XIII.

Morkūnaitė V, Baranauskienė L, Zubrienė A, Kairys V, Ivanova J, Trapencieris P, Matulis D. Morkūnaitė V, et al. Among authors: trapencieris p. Biomed Res Int. 2014;2014:638902. doi: 10.1155/2014/638902. Epub 2014 Sep 3. Biomed Res Int. 2014. PMID: 25276805 Free PMC article.

7

A Novel Aziridine-based Bruton's Tyrosine Kinase Inhibitor Induces Apoptosis Through Down-regulation of p65/RelA Phosphorylation on Serine 536 and ERK1/2 in Mantle Cell Lymphoma.

Romanchikova N, Strods A, Strazdina J, Strumfs B, Trapencieris P. Romanchikova N, et al. Among authors: trapencieris p. Anticancer Res. 2016 Nov;36(11):6133-6140. doi: 10.21873/anticanres.11204. Anticancer Res. 2016. PMID: 27793942

8

3-Arylaziridine-2-carboxylic Acid Derivatives and (3-Arylaziridin-2-yl)ketones: The Aziridination Approaches.

Strumfs B, Uljanovs R, Velikijs K, Trapencieris P, Strumfa I. Strumfs B, et al. Among authors: trapencieris p. Int J Mol Sci. 2021 Sep 13;22(18):9861. doi: 10.3390/ijms22189861. Int J Mol Sci. 2021. PMID: 34576025 Free PMC article. Review.

9

Wedelolactone Targets EZH2-mediated Histone H3K27 Methylation in Mantle Cell Lymphoma.

Romanchikova N, Trapencieris P. Romanchikova N, et al. Among authors: trapencieris p. Anticancer Res. 2019 Aug;39(8):4179-4184. doi: 10.21873/anticanres.13577. Anticancer Res. 2019. PMID: 31366503

10

Plasmepsin inhibitory activity and structure-guided optimization of a potent hydroxyethylamine-based antimalarial hit.

Jaudzems K, Tars K, Maurops G, Ivdra N, Otikovs M, Leitans J, Kanepe-Lapsa I, Domraceva I, Mutule I, Trapencieris P, Blackman MJ, Jirgensons A. Jaudzems K, et al. Among authors: trapencieris p. ACS Med Chem Lett. 2014 Jan 13;5(4):373-7. doi: 10.1021/ml4004952. eCollection 2014 Apr 10. ACS Med Chem Lett. 2014. PMID: 24900843 Free PMC article.

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