Buckner FS - Search Results

1

Phenotypic Drug Discovery for Human African Trypanosomiasis: A Powerful Approach.

Buckner FS, Buchynskyy A, Nagendar P, Patrick DA, Gillespie JR, Herbst Z, Tidwell RR, Gelb MH. Buckner FS, et al. Trop Med Infect Dis. 2020 Feb 5;5(1):23. doi: 10.3390/tropicalmed5010023. Trop Med Infect Dis. 2020. PMID: 32033395 Free PMC article.

2

Urea Derivatives of 2-Aryl-benzothiazol-5-amines: A New Class of Potential Drugs for Human African Trypanosomiasis.

Patrick DA, Gillespie JR, McQueen J, Hulverson MA, Ranade RM, Creason SA, Herbst ZM, Gelb MH, Buckner FS, Tidwell RR. Patrick DA, et al. Among authors: buckner fs. J Med Chem. 2017 Feb 9;60(3):957-971. doi: 10.1021/acs.jmedchem.6b01163. Epub 2016 Dec 19. J Med Chem. 2017. PMID: 27992217 Free PMC article.

3

Protein farnesyl transferase inhibitors for the treatment of malaria and African trypanosomiasis.

Buckner FS, Eastman RT, Yokoyama K, Gelb MH, Van Voorhis WC. Buckner FS, et al. Curr Opin Investig Drugs. 2005 Aug;6(8):791-7. Curr Opin Investig Drugs. 2005. PMID: 16121685 Review.

4

Glycogen synthase kinase 3 is a potential drug target for African trypanosomiasis therapy.

Ojo KK, Gillespie JR, Riechers AJ, Napuli AJ, Verlinde CL, Buckner FS, Gelb MH, Domostoj MM, Wells SJ, Scheer A, Wells TN, Van Voorhis WC. Ojo KK, et al. Among authors: buckner fs. Antimicrob Agents Chemother. 2008 Oct;52(10):3710-7. doi: 10.1128/AAC.00364-08. Epub 2008 Jul 21. Antimicrob Agents Chemother. 2008. PMID: 18644955 Free PMC article.

5

Substituted 2-phenylimidazopyridines: a new class of drug leads for human African trypanosomiasis.

Tatipaka HB, Gillespie JR, Chatterjee AK, Norcross NR, Hulverson MA, Ranade RM, Nagendar P, Creason SA, McQueen J, Duster NA, Nagle A, Supek F, Molteni V, Wenzler T, Brun R, Glynne R, Buckner FS, Gelb MH. Tatipaka HB, et al. Among authors: buckner fs. J Med Chem. 2014 Feb 13;57(3):828-35. doi: 10.1021/jm401178t. Epub 2014 Jan 15. J Med Chem. 2014. PMID: 24354316 Free PMC article.

6

Discovery of N-(2-aminoethyl)-N-benzyloxyphenyl benzamides: New potent Trypanosoma brucei inhibitors.

Buchynskyy A, Gillespie JR, Hulverson MA, McQueen J, Creason SA, Ranade RM, Duster NA, Gelb MH, Buckner FS. Buchynskyy A, et al. Among authors: buckner fs. Bioorg Med Chem. 2017 Mar 1;25(5):1571-1584. doi: 10.1016/j.bmc.2016.11.019. Epub 2016 Nov 12. Bioorg Med Chem. 2017. PMID: 28187957 Free PMC article.

7

1-Benzyl-3-aryl-2-thiohydantoin Derivatives as New Anti-Trypanosoma brucei Agents: SAR and in Vivo Efficacy.

Buchynskyy A, Gillespie JR, Herbst ZM, Ranade RM, Buckner FS, Gelb MH. Buchynskyy A, et al. Among authors: buckner fs. ACS Med Chem Lett. 2017 Jul 10;8(8):886-891. doi: 10.1021/acsmedchemlett.7b00230. eCollection 2017 Aug 10. ACS Med Chem Lett. 2017. PMID: 28835807 Free PMC article.

8

Triazolopyrimidines and Imidazopyridines: Structure-Activity Relationships and in Vivo Efficacy for Trypanosomiasis.

Nagendar P, Gillespie JR, Herbst ZM, Ranade RM, Molasky NMR, Faghih O, Turner RM, Gelb MH, Buckner FS. Nagendar P, et al. Among authors: buckner fs. ACS Med Chem Lett. 2018 Dec 4;10(1):105-110. doi: 10.1021/acsmedchemlett.8b00498. eCollection 2019 Jan 10. ACS Med Chem Lett. 2018. PMID: 30655955 Free PMC article.

9

Early Stages of Drug Discovery in an Academic Institution and Involvement of Pharma for Advancing Promising Leads.

Gelb MH, Buckner FS. Gelb MH, et al. Among authors: buckner fs. ACS Infect Dis. 2021 Jul 9;7(7):1874-1876. doi: 10.1021/acsinfecdis.1c00091. Epub 2021 Apr 19. ACS Infect Dis. 2021. PMID: 33871981 Free PMC article.

10

Rational modification of a candidate cancer drug for use against Chagas disease.

Kraus JM, Verlinde CL, Karimi M, Lepesheva GI, Gelb MH, Buckner FS. Kraus JM, et al. Among authors: buckner fs. J Med Chem. 2009 Mar 26;52(6):1639-47. doi: 10.1021/jm801313t. J Med Chem. 2009. PMID: 19239254 Free PMC article.

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