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Improved translation of stability for conjugated antibodies using an in vitro whole blood assay.
MAbs. 2020 Jan-Dec;12(1):1715705. doi: 10.1080/19420862.2020.1715705.
MAbs. 2020.
PMID: 31997712
Free PMC article.
Characterizing and Quantitating Therapeutic Tethered Multimeric Antibody Degradation Using Affinity Capture Mass Spectrometry.
Li W, Srikumar N, Forrest WF, Ellerman D, Gu C, Tchelepi R, Lazar GA, Liu Y, Tran JC.
Li W, et al. Among authors: tchelepi r.
Anal Chem. 2020 May 19;92(10):6839-6843. doi: 10.1021/acs.analchem.9b05739. Epub 2020 May 4.
Anal Chem. 2020.
PMID: 32309925
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Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates.
Nicolaou KC, Li R, Chen Q, Lu Z, Pitsinos EN, Schammel A, Lin B, Gu C, Sarvaiya H, Tchelepi R, Valdiosera A, Clubb J, Barbour N, Sisodiya V, Sandoval J, Lee C, Aujay M, Gavrilyuk J.
Nicolaou KC, et al. Among authors: tchelepi r.
J Am Chem Soc. 2020 Jul 22;142(29):12890-12899. doi: 10.1021/jacs.0c06554. Epub 2020 Jul 14.
J Am Chem Soc. 2020.
PMID: 32662641
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Synthesis and Comparative In Vivo Evaluation of Site-Specifically Labeled Radioimmunoconjugates for DLL3-Targeted ImmunoPET.
Sharma SK, Adumeau P, Keinänen O, Sisodiya V, Sarvaiya H, Tchelepi R, Korsen JA, Pourat J, Edwards KJ, Ragupathi A, Hamdy O, Saunders LR, Rudin CM, Poirier JT, Lewis JS, Zeglis BM.
Sharma SK, et al. Among authors: tchelepi r.
Bioconjug Chem. 2021 Jul 21;32(7):1255-1262. doi: 10.1021/acs.bioconjchem.1c00121. Epub 2021 Apr 9.
Bioconjug Chem. 2021.
PMID: 33835770
Free PMC article.
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Evaluation of PNU-159682 antibody drug conjugates (ADCs).
Holte D, Lyssikatos JP, Valdiosera AM, Swinney Z, Sisodiya V, Sandoval J, Lee C, Aujay MA, Tchelepi RB, Hamdy OM, Gu C, Lin B, Sarvaiya H, Pysz MA, Laysang A, Williams S, Jun Lee D, Holda MK, Purcell JW, Gavrilyuk J.
Holte D, et al. Among authors: tchelepi rb.
Bioorg Med Chem Lett. 2020 Dec 15;30(24):127640. doi: 10.1016/j.bmcl.2020.127640. Epub 2020 Oct 28.
Bioorg Med Chem Lett. 2020.
PMID: 33127540
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