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Trifluoromethyl Dihydrothiazine-Based β-Secretase (BACE1) Inhibitors with Robust Central β-Amyloid Reduction and Minimal Covalent Binding Burden.
Anan K, Iso Y, Oguma T, Nakahara K, Suzuki S, Yamamoto T, Matsuoka E, Ito H, Sakaguchi G, Ando S, Morimoto K, Kanegawa N, Kido Y, Kawachi T, Fukushima T, Teisman A, Urmaliya V, Dhuyvetter D, Borghys H, Austin N, Van Den Bergh A, Verboven P, Bischoff F, Gijsen HJM, Yamano Y, Kusakabe K. Anan K, et al. Among authors: kawachi t. ChemMedChem. 2019 Nov 20;14(22):1894-1910. doi: 10.1002/cmdc.201900478. Epub 2019 Nov 12. ChemMedChem. 2019. PMID: 31657130
Discovery of 2-Sulfinyl-Diazabicyclooctane Derivatives, Potential Oral β-Lactamase Inhibitors for Infections Caused by Serine β-Lactamase-Producing Enterobacterales.
Fujiu M, Yokoo K, Sato J, Shibuya S, Komano K, Kusano H, Sato S, Aoki T, Kohira N, Kanazawa S, Watari R, Kawachi T, Hirakawa Y, Nagamatsu D, Kashiwagi E, Maki H, Yamawaki K. Fujiu M, et al. Among authors: kawachi t. J Med Chem. 2021 Jul 8;64(13):9496-9512. doi: 10.1021/acs.jmedchem.1c00799. Epub 2021 Jun 18. J Med Chem. 2021. PMID: 34143627
Introduction of a Thio Functional Group to Diazabicyclooctane: An Effective Modification to Potentiate the Activity of β-Lactams against Gram-Negative Bacteria Producing Class A, C, and D Serine β-Lactamases.
Fujiu M, Yokoo K, Sato J, Shibuya S, Komano K, Kusano H, Sato S, Aoki T, Kohira N, Miyagawa S, Kawachi T, Yamawaki K. Fujiu M, et al. Among authors: kawachi t. ACS Infect Dis. 2020 Nov 13;6(11):3034-3047. doi: 10.1021/acsinfecdis.0c00560. Epub 2020 Nov 4. ACS Infect Dis. 2020. PMID: 33147950
Damage threshold of LiF crystal irradiated by femtosecond hard XFEL pulse sequence.
Makarov S, Grigoryev S, Inogamov N, Filippov E, Pikuz T, Ozaki N, Ishino M, Nishikino M, Dinh TH, Kawachi T, Zanaveskin M, Makita M, Nakatsutsumi M, Preston TR, Appel K, Konopkova Z, Cerantola V, Brambrink E, Schwinkendorf JP, Mohacsi I, Vozda V, Hajkova V, Burian T, Chalupsky J, Juha L, Zhakhovsky V, Zastrau U, Pikuz S. Makarov S, et al. Among authors: kawachi t. Opt Express. 2023 Jul 31;31(16):26383-26397. doi: 10.1364/OE.486868. Opt Express. 2023. PMID: 37710501 Free article.
229 results