Kongstad KT - Search Results

1

Developing New 4-PIOL and 4-PHP Analogues for Photoinactivation of γ-Aminobutyric Acid Type A Receptors.

Mortensen M, Krall J, Kongstad KT, Brygger BM, Lenzi O, Francotte P, Sørensen TE, Nielsen B, Jensen AA, Smart TG, Frølund B. Mortensen M, et al. Among authors: kongstad kt. ACS Chem Neurosci. 2019 Nov 20;10(11):4669-4684. doi: 10.1021/acschemneuro.9b00478. Epub 2019 Oct 21. ACS Chem Neurosci. 2019. PMID: 31589403

2

5-(Piperidin-4-yl)-3-hydroxypyrazole: A novel scaffold for probing the orthosteric γ-aminobutyric acid type A receptor binding site.

Krall J, Kongstad KT, Nielsen B, Sørensen TE, Balle T, Jensen AA, Frølund B. Krall J, et al. Among authors: kongstad kt. ChemMedChem. 2014 Nov;9(11):2475-85. doi: 10.1002/cmdc.201402248. Epub 2014 Aug 26. ChemMedChem. 2014. PMID: 25156407

3

Discovery of 2-(Imidazo[1,2- b]pyridazin-2-yl)acetic Acid as a New Class of Ligands Selective for the γ-Hydroxybutyric Acid (GHB) High-Affinity Binding Sites.

Krall J, Bavo F, Falk-Petersen CB, Jensen CH, Nielsen JO, Tian Y, Anglani V, Kongstad KT, Piilgaard L, Nielsen B, Gloriam DE, Kehler J, Jensen AA, Harpsøe K, Wellendorph P, Frølund B. Krall J, et al. Among authors: kongstad kt. J Med Chem. 2019 Mar 14;62(5):2798-2813. doi: 10.1021/acs.jmedchem.9b00131. Epub 2019 Feb 27. J Med Chem. 2019. PMID: 30763084

4

Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at γ-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters.

Giraudo A, Krall J, Bavo F, Nielsen B, Kongstad KT, Rolando B, De Blasio R, Gloriam DE, Löffler R, Thiesen L, Harpsøe K, Frydenvang K, Boschi D, Wellendorph P, Lolli ML, Jensen AA, Frølund B. Giraudo A, et al. Among authors: kongstad kt. J Med Chem. 2019 Jun 27;62(12):5797-5809. doi: 10.1021/acs.jmedchem.9b00026. Epub 2019 Jun 5. J Med Chem. 2019. PMID: 31117514 Free article.

5

4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site.

Giraudo A, Krall J, Nielsen B, Sørensen TE, Kongstad KT, Rolando B, Boschi D, Frølund B, Lolli ML. Giraudo A, et al. Among authors: kongstad kt. Eur J Med Chem. 2018 Oct 5;158:311-321. doi: 10.1016/j.ejmech.2018.08.094. Epub 2018 Sep 5. Eur J Med Chem. 2018. PMID: 30223119 Free article.

6

Molecular Hybridization of Potent and Selective γ-Hydroxybutyric Acid (GHB) Ligands: Design, Synthesis, Binding Studies, and Molecular Modeling of Novel 3-Hydroxycyclopent-1-enecarboxylic Acid (HOCPCA) and trans-γ-Hydroxycrotonic Acid (T-HCA) Analogs.

Krall J, Jensen CH, Bavo F, Falk-Petersen CB, Haugaard AS, Vogensen SB, Tian Y, Nittegaard-Nielsen M, Sigurdardóttir SB, Kehler J, Kongstad KT, Gloriam DE, Clausen RP, Harpsøe K, Wellendorph P, Frølund B. Krall J, et al. Among authors: kongstad kt. J Med Chem. 2017 Nov 9;60(21):9022-9039. doi: 10.1021/acs.jmedchem.7b01351. Epub 2017 Oct 30. J Med Chem. 2017. PMID: 29028338

7

Positive allosteric modulation of the GHB high-affinity binding site by the GABAA receptor modulator monastrol and the flavonoid catechin.

Eghorn LF, Hoestgaard-Jensen K, Kongstad KT, Bay T, Higgins D, Frølund B, Wellendorph P. Eghorn LF, et al. Among authors: kongstad kt. Eur J Pharmacol. 2014 Oct 5;740:570-7. doi: 10.1016/j.ejphar.2014.06.028. Epub 2014 Jun 25. Eur J Pharmacol. 2014. PMID: 24973695

8

¹⁹F-substituted amino acids as an alternative to fluorophore labels: monitoring of degradation and cellular uptake of analogues of penetratin by ¹⁹F NMR.

Christensen MV, Kongstad KT, Sondergaard TE, Staerk D, Nielsen HM, Franzyk H, Wimmer R. Christensen MV, et al. Among authors: kongstad kt. J Biomol NMR. 2019 Apr;73(3-4):167-182. doi: 10.1007/s10858-019-00239-3. Epub 2019 Mar 18. J Biomol NMR. 2019. PMID: 30887171

9

Potential of Polygonum cuspidatum Root as an Antidiabetic Food: Dual High-Resolution α-Glucosidase and PTP1B Inhibition Profiling Combined with HPLC-HRMS and NMR for Identification of Antidiabetic Constituents.

Zhao Y, Chen MX, Kongstad KT, Jäger AK, Staerk D. Zhao Y, et al. Among authors: kongstad kt. J Agric Food Chem. 2017 Jun 7;65(22):4421-4427. doi: 10.1021/acs.jafc.7b01353. Epub 2017 May 24. J Agric Food Chem. 2017. PMID: 28497962

10

Unraveling the complexity of complex mixtures by combining high-resolution pharmacological, analytical and spectroscopic techniques: antidiabetic constituents in Chinese medicinal plants.

Zhao Y, Kongstad KT, Liu Y, He C, Staerk D. Zhao Y, et al. Among authors: kongstad kt. Faraday Discuss. 2019 Aug 15;218(0):202-218. doi: 10.1039/c8fd00223a. Faraday Discuss. 2019. PMID: 31119225

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