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Tacrine-O-protected phenolics heterodimers as multitarget-directed ligands against Alzheimer's disease: Selective subnanomolar BuChE inhibitors.
Eur J Med Chem. 2019 Nov 1;181:111550. doi: 10.1016/j.ejmech.2019.07.053. Epub 2019 Jul 22.
Eur J Med Chem. 2019.
PMID: 31376562
New tacrine dimers with antioxidant linkers as dual drugs: Anti-Alzheimer's and antiproliferative agents.
Roldán-Peña JM, Alejandre-Ramos D, López Ó, Maya I, Lagunes I, Padrón JM, Peña-Altamira LE, Bartolini M, Monti B, Bolognesi ML, Fernández-Bolaños JG.
Roldán-Peña JM, et al.
Eur J Med Chem. 2017 Sep 29;138:761-773. doi: 10.1016/j.ejmech.2017.06.048. Epub 2017 Jun 27.
Eur J Med Chem. 2017.
PMID: 28728108
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Biotinylated selenocyanates: Potent and selective cytostatic agents.
Roldán-Peña JM, Puerta A, Dinić J, Jovanović Stojanov S, González-Bakker A, Hicke FJ, Mishra A, Piyasaengthong A, Maya I, Walton JW, Pešić M, Padrón JM, Fernández-Bolaños JG, López Ó.
Roldán-Peña JM, et al.
Bioorg Chem. 2023 Apr;133:106410. doi: 10.1016/j.bioorg.2023.106410. Epub 2023 Feb 8.
Bioorg Chem. 2023.
PMID: 36822000
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