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2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials.
Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Ayginin AA, Skvortsov DA, Komarova KS, Sadovnikov SV, Matniyazov R, Sofronova AA, Malyshev AS, Machulkin AE, Petrov RA, Lukianov D, Iarovenko S, Bezrukov DS, Baymiev AK, Dontsova OA. Ivanenkov YA, et al. J Antibiot (Tokyo). 2019 Nov;72(11):827-833. doi: 10.1038/s41429-019-0211-y. Epub 2019 Jul 29. J Antibiot (Tokyo). 2019. PMID: 31358913
Novel oral anti-influenza drug candidate AV5080.
Ivachtchenko AV, Ivanenkov YA, Mitkin OD, Yamanushkin PM, Bichko VV, Shevkun NA, Karapetian RN, Leneva IA, Borisova OV, Veselov MS. Ivachtchenko AV, et al. Among authors: ivanenkov ya. J Antimicrob Chemother. 2014 Jul;69(7):1892-902. doi: 10.1093/jac/dku074. Epub 2014 Apr 11. J Antimicrob Chemother. 2014. PMID: 24729605
Design, synthesis and biological evaluation of novel potent MDM2/p53 small-molecule inhibitors.
Ivanenkov YA, Vasilevski SV, Beloglazkina EK, Kukushkin ME, Machulkin AE, Veselov MS, Chufarova NV, Chernyaginab ES, Vanzcool AS, Zyk NV, Skvortsov DA, Khutornenko AA, Rusanov AL, Tonevitsky AG, Dontsova OA, Majouga AG. Ivanenkov YA, et al. Bioorg Med Chem Lett. 2015 Jan 15;25(2):404-9. doi: 10.1016/j.bmcl.2014.09.070. Epub 2014 Oct 2. Bioorg Med Chem Lett. 2015. PMID: 25479770
Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists.
Ivachtchenko AV, Ivanenkov YA, Mitkin OD, Vorobiev AA, Kuznetsova IV, Shevkun NA, Koryakova AG, Karapetian RN, Trifelenkov AS, Kravchenko DV, Veselov MS, Chufarova NV. Ivachtchenko AV, et al. Among authors: ivanenkov ya. Eur J Med Chem. 2015 Jun 24;99:51-66. doi: 10.1016/j.ejmech.2015.05.039. Epub 2015 Jun 2. Eur J Med Chem. 2015. PMID: 26046313
In Silico Approaches to the Design of NS5A Inhibitors.
Ivanenkov YA, Veselov MS, Aladinskiy VA, Shakhbazyan AG, Yartseva SM, Majouga AG, Aladinskaya AV, Vantskul AS, Leonov SV, Ivachtchenko AV, Koteliansky VE. Ivanenkov YA, et al. Curr Top Med Chem. 2016;16(12):1383-91. doi: 10.2174/1568026616666151120113705. Curr Top Med Chem. 2016. PMID: 26585932 Review.
Computational insight into the chemical space of plant growth regulators.
Bushkov NA, Veselov MS, Chuprov-Netochin RN, Marusich EI, Majouga AG, Volynchuk PB, Shumilina DV, Leonov SV, Ivanenkov YA. Bushkov NA, et al. Among authors: ivanenkov ya. Phytochemistry. 2016 Feb;122:254-264. doi: 10.1016/j.phytochem.2015.12.006. Epub 2015 Dec 23. Phytochemistry. 2016. PMID: 26723884
Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivatives.
Ivanenkov YA, Veselov MS, Rezekin IG, Skvortsov DA, Sandulenko YB, Polyakova MV, Bezrukov DS, Vasilevsky SV, Kukushkin ME, Moiseeva AA, Finko AV, Koteliansky VE, Klyachko NL, Filatova LA, Beloglazkina EK, Zyk NV, Majouga AG. Ivanenkov YA, et al. Bioorg Med Chem. 2016 Feb 15;24(4):802-11. doi: 10.1016/j.bmc.2015.12.050. Epub 2016 Jan 2. Bioorg Med Chem. 2016. PMID: 26780833
85 results