Jorda R - Search Results

1

Tetrahydropyrazolo[1,5-a]pyridine-fused steroids and their in vitro biological evaluation in prostate cancer.

Jorda R, Lopes SMM, Řezníčková E, Ajani H, Pereira AV, Gomes CSB, M V D Pinho E Melo T. Jorda R, et al. Eur J Med Chem. 2019 Sep 15;178:168-176. doi: 10.1016/j.ejmech.2019.05.064. Epub 2019 May 30. Eur J Med Chem. 2019. PMID: 31181481

2

Pyrazolo[4,3-d]pyrimidine bioisostere of roscovitine: evaluation of a novel selective inhibitor of cyclin-dependent kinases with antiproliferative activity.

Jorda R, Havlícek L, McNae IW, Walkinshaw MD, Voller J, Sturc A, Navrátilová J, Kuzma M, Mistrík M, Bártek J, Strnad M, Krystof V. Jorda R, et al. J Med Chem. 2011 Apr 28;54(8):2980-93. doi: 10.1021/jm200064p. Epub 2011 Apr 6. J Med Chem. 2011. PMID: 21417417

3

The selective P-TEFb inhibitor CAN508 targets angiogenesis.

Kryštof V, Rárová L, Liebl J, Zahler S, Jorda R, Voller J, Cankař P. Kryštof V, et al. Among authors: jorda r. Eur J Med Chem. 2011 Sep;46(9):4289-94. doi: 10.1016/j.ejmech.2011.06.035. Epub 2011 Jul 3. Eur J Med Chem. 2011. PMID: 21777997

4

Synthesis and in vitro biological evaluation of 2,6,9-trisubstituted purines targeting multiple cyclin-dependent kinases.

Zatloukal M, Jorda R, Gucký T, Řezníčková E, Voller J, Pospíšil T, Malínková V, Adamcová H, Kryštof V, Strnad M. Zatloukal M, et al. Among authors: jorda r. Eur J Med Chem. 2013 Mar;61:61-72. doi: 10.1016/j.ejmech.2012.06.036. Epub 2012 Jun 23. Eur J Med Chem. 2013. PMID: 22770608

5

A novel series of highly potent 2,6,9-trisubstituted purine cyclin-dependent kinase inhibitors.

Gucký T, Jorda R, Zatloukal M, Bazgier V, Berka K, Řezníčková E, Béres T, Strnad M, Kryštof V. Gucký T, et al. Among authors: jorda r. J Med Chem. 2013 Aug 8;56(15):6234-47. doi: 10.1021/jm4006884. Epub 2013 Jul 24. J Med Chem. 2013. PMID: 23829517

6

Substituted 2-hydroxy-N-(arylalkyl)benzamides induce apoptosis in cancer cell lines.

Imramovský A, Jorda R, Pauk K, Rezníčková E, Dušek J, Hanusek J, Kryštof V. Imramovský A, et al. Among authors: jorda r. Eur J Med Chem. 2013 Oct;68:253-9. doi: 10.1016/j.ejmech.2013.08.009. Epub 2013 Aug 14. Eur J Med Chem. 2013. PMID: 23981532

7

Novel arylazopyrazole inhibitors of cyclin-dependent kinases.

Jorda R, Schütznerová E, Cankař P, Brychtová V, Navrátilová J, Kryštof V. Jorda R, et al. Bioorg Med Chem. 2015 May 1;23(9):1975-81. doi: 10.1016/j.bmc.2015.03.025. Epub 2015 Mar 14. Bioorg Med Chem. 2015. PMID: 25835357

8

2,6,9-Trisubstituted purines as CRK3 kinase inhibitors with antileishmanial activity in vitro.

Řezníčková E, Popa A, Gucký T, Zatloukal M, Havlíček L, Bazgier V, Berka K, Jorda R, Popa I, Nasereddin A, Jaffe CL, Kryštof V, Strnad M. Řezníčková E, et al. Among authors: jorda r. Bioorg Med Chem Lett. 2015 Jun 1;25(11):2298-301. doi: 10.1016/j.bmcl.2015.04.030. Epub 2015 Apr 16. Bioorg Med Chem Lett. 2015. PMID: 25937014

9

Characterization of a Pyrazolo[4,3-d]pyrimidine Inhibitor of Cyclin-Dependent Kinases 2 and 5 and Aurora A With Pro-Apoptotic and Anti-Angiogenic Activity In Vitro.

Řezníčková E, Weitensteiner S, Havlíček L, Jorda R, Gucký T, Berka K, Bazgier V, Zahler S, Kryštof V, Strnad M. Řezníčková E, et al. Among authors: jorda r. Chem Biol Drug Des. 2015 Dec;86(6):1528-40. doi: 10.1111/cbdd.12618. Epub 2015 Sep 16. Chem Biol Drug Des. 2015. PMID: 26198005

10

Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors.

Baltus CB, Jorda R, Marot C, Berka K, Bazgier V, Kryštof V, Prié G, Viaud-Massuard MC. Baltus CB, et al. Among authors: jorda r. Eur J Med Chem. 2016 Jan 27;108:701-719. doi: 10.1016/j.ejmech.2015.12.023. Epub 2015 Dec 19. Eur J Med Chem. 2016. PMID: 26741853

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