Kołaczkowski M - Search Results

1

Anti-Alzheimer's multitarget-directed ligands with serotonin 5-HT₆ antagonist, butyrylcholinesterase inhibitory, and antioxidant activity.

Marcinkowska M, Bucki A, Panek D, Siwek A, Fajkis N, Bednarski M, Zygmunt M, Godyń J, Del Rio Valdivieso A, Kotańska M, Kołaczkowski M, Więckowska A. Marcinkowska M, et al. Among authors: kolaczkowski m. Arch Pharm (Weinheim). 2019 Jul;352(7):e1900041. doi: 10.1002/ardp.201900041. Epub 2019 Jun 4. Arch Pharm (Weinheim). 2019. PMID: 31162703

2

Novel mannich bases, 5-arylimidazolidine-2,4-dione derivatives with dual 5-HT(1A) receptor and serotonin transporter affinity.

Czopek A, Kołaczkowski M, Bucki A, Byrtus H, Pawłowski M, Siwek A, Bojarski AJ, Bednarski M, Wróbel D, Wesołowska A. Czopek A, et al. Among authors: kolaczkowski m. Arch Pharm (Weinheim). 2013 Feb;346(2):98-109. doi: 10.1002/ardp.201200378. Epub 2013 Jan 3. Arch Pharm (Weinheim). 2013. PMID: 23288448

3

Ligand-optimized homology models of D₁ and D₂ dopamine receptors: application for virtual screening.

Kołaczkowski M, Bucki A, Feder M, Pawłowski M. Kołaczkowski M, et al. J Chem Inf Model. 2013 Mar 25;53(3):638-48. doi: 10.1021/ci300413h. Epub 2013 Feb 27. J Chem Inf Model. 2013. PMID: 23398329

4

Partial agonist efficacy of EMD386088, a 5-HT6 receptor ligand, in functional in vitro assays.

Jastrzębska-Więsek M, Siwek A, Kazek G, Nawieśniak B, Partyka A, Marcinkowska M, Kołaczkowski M, Wesołowska A. Jastrzębska-Więsek M, et al. Among authors: kolaczkowski m. Pharmacol Rep. 2013;65(4):998-1005. doi: 10.1016/s1734-1140(13)71081-8. Pharmacol Rep. 2013. PMID: 24145094 Free article.

5

Novel arylsulfonamide derivatives with 5-HT₆/5-HT₇ receptor antagonism targeting behavioral and psychological symptoms of dementia.

Kołaczkowski M, Marcinkowska M, Bucki A, Pawłowski M, Mitka K, Jaśkowska J, Kowalski P, Kazek G, Siwek A, Wasik A, Wesołowska A, Mierzejewski P, Bienkowski P. Kołaczkowski M, et al. J Med Chem. 2014 Jun 12;57(11):4543-57. doi: 10.1021/jm401895u. Epub 2014 May 23. J Med Chem. 2014. PMID: 24805037

6

Pharmacological evaluation of the anxiolytic-like effects of EMD 386088, a partial 5-HT6 receptor agonist, in the rat elevated plus-maze and Vogel conflict tests.

Jastrzębska-Więsek M, Siwek A, Partyka A, Kubacka M, Mogilski S, Wasik A, Kołaczkowski M, Wesołowska A. Jastrzębska-Więsek M, et al. Among authors: kolaczkowski m. Neuropharmacology. 2014 Oct;85:253-62. doi: 10.1016/j.neuropharm.2014.05.036. Epub 2014 Jun 4. Neuropharmacology. 2014. PMID: 24905144

7

Studies on the anticonvulsant activity and influence on GABA-ergic neurotransmission of 1,2,4-triazole-3-thione- based compounds.

Plech T, Kaproń B, Luszczki JJ, Wujec M, Paneth A, Siwek A, Kołaczkowski M, Zołnierek M, Nowak G. Plech T, et al. Among authors: kolaczkowski m. Molecules. 2014 Jul 31;19(8):11279-99. doi: 10.3390/molecules190811279. Molecules. 2014. PMID: 25090118 Free PMC article.

8

Studies on the anticonvulsant activity of 4-alkyl-1,2,4-triazole-3-thiones and their effect on GABAergic system.

Plech T, Kaproń B, Luszczki JJ, Paneth A, Siwek A, Kołaczkowski M, Żołnierek M, Nowak G. Plech T, et al. Among authors: kolaczkowski m. Eur J Med Chem. 2014 Oct 30;86:690-9. doi: 10.1016/j.ejmech.2014.09.034. Epub 2014 Sep 16. Eur J Med Chem. 2014. PMID: 25226229

9

Antidepressant- and anxiolytic-like activity of 7-phenylpiperazinylalkyl-1,3-dimethyl-purine-2,6-dione derivatives with diversified 5-HT₁A receptor functional profile.

Partyka A, Chłoń-Rzepa G, Wasik A, Jastrzębska-Więsek M, Bucki A, Kołaczkowski M, Satała G, Bojarski AJ, Wesołowska A. Partyka A, et al. Among authors: kolaczkowski m. Bioorg Med Chem. 2015 Jan 1;23(1):212-21. doi: 10.1016/j.bmc.2014.11.008. Epub 2014 Nov 11. Bioorg Med Chem. 2015. PMID: 25435254

10

Novel 5-HT6 receptor antagonists/D2 receptor partial agonists targeting behavioral and psychological symptoms of dementia.

Kołaczkowski M, Marcinkowska M, Bucki A, Śniecikowska J, Pawłowski M, Kazek G, Siwek A, Jastrzębska-Więsek M, Partyka A, Wasik A, Wesołowska A, Mierzejewski P, Bienkowski P. Kołaczkowski M, et al. Eur J Med Chem. 2015 Mar 6;92:221-35. doi: 10.1016/j.ejmech.2014.12.045. Epub 2014 Dec 24. Eur J Med Chem. 2015. PMID: 25557493

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