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Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening.
J Am Chem Soc. 2019 Jun 5;141(22):8951-8968. doi: 10.1021/jacs.9b02822. Epub 2019 May 22.
J Am Chem Soc. 2019.
PMID: 31060360
Free PMC article.
Novel Starting Points for Human Glycolate Oxidase Inhibitors, Revealed by Crystallography-Based Fragment Screening.
Mackinnon SR, Bezerra GA, Krojer T, Szommer T, von Delft F, Brennan PE, Yue WW.
Mackinnon SR, et al. Among authors: szommer t.
Front Chem. 2022 May 4;10:844598. doi: 10.3389/fchem.2022.844598. eCollection 2022.
Front Chem. 2022.
PMID: 35601556
Free PMC article.
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Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7.
Gerken PA, Wolstenhulme JR, Tumber A, Hatch SB, Zhang Y, Müller S, Chandler SA, Mair B, Li F, Nijman SMB, Konietzny R, Szommer T, Yapp C, Fedorov O, Benesch JLP, Vedadi M, Kessler BM, Kawamura A, Brennan PE, Smith MD.
Gerken PA, et al. Among authors: szommer t.
Angew Chem Int Ed Engl. 2017 Dec 4;56(49):15555-15559. doi: 10.1002/anie.201706788. Epub 2017 Nov 7.
Angew Chem Int Ed Engl. 2017.
PMID: 28976073
Free PMC article.
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Inhibition of Histone H3K27 Demethylases Inactivates Brachyury (TBXT) and Promotes Chordoma Cell Death.
Cottone L, Cribbs AP, Khandelwal G, Wells G, Ligammari L, Philpott M, Tumber A, Lombard P, Hookway ES, Szommer T, Johansson C, Brennan PE, Pillay N, Jenner RG, Oppermann U, Flanagan AM.
Cottone L, et al. Among authors: szommer t.
Cancer Res. 2020 Oct 15;80(20):4540-4551. doi: 10.1158/0008-5472.CAN-20-1387. Epub 2020 Aug 27.
Cancer Res. 2020.
PMID: 32855205
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Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist.
Balıkçı E, Marques AMC, Bauer LG, Seupel R, Bennett J, Raux B, Buchan K, Simelis K, Singh U, Rogers C, Ward J, Cheng C, Szommer T, Schützenhofer K, Elkins JM, Sloman DL, Ahel I, Fedorov O, Brennan PE, Huber KVM.
Balıkçı E, et al. Among authors: szommer t.
J Med Chem. 2024 May 9;67(9):7245-7259. doi: 10.1021/acs.jmedchem.4c00072. Epub 2024 Apr 18.
J Med Chem. 2024.
PMID: 38635563
Free PMC article.
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Parallel synthesis of 1,2,4-triazole derivatives using microwave and continuous-flow techniques.
Szommer T, Lukács A, Kovács J, Szabó MJ, Hoffmann MG, Schmitt MH, Gerencsér J.
Szommer T, et al.
Mol Divers. 2012 Feb;16(1):81-90. doi: 10.1007/s11030-012-9357-2. Epub 2012 Jan 26.
Mol Divers. 2012.
PMID: 22278610
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Enhanced hit-to-lead process using bioanalogous lead evolution and chemogenomics: application in designing selective matrix metalloprotease inhibitors.
Papp A, Szommer T, Barna L, Gyimesi G, Ferdinandy P, Spadoni C, Darvas F, Fujita T, Urge L, Dormán G.
Papp A, et al. Among authors: szommer t.
Expert Opin Drug Discov. 2007 May;2(5):707-23. doi: 10.1517/17460441.2.5.707.
Expert Opin Drug Discov. 2007.
PMID: 23488960
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