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Quorum Sensing as Antivirulence Target in Cystic Fibrosis Pathogens.
Scoffone VC, Trespidi G, Chiarelli LR, Barbieri G, Buroni S. Scoffone VC, et al. Among authors: chiarelli lr. Int J Mol Sci. 2019 Apr 13;20(8):1838. doi: 10.3390/ijms20081838. Int J Mol Sci. 2019. PMID: 31013936 Free PMC article. Review.
Targeting Siderophore-Mediated Iron Uptake in M. abscessus: A New Strategy to Limit the Virulence of Non-Tuberculous Mycobacteria.
Mori M, Stelitano G, Cazzaniga G, Gelain A, Tresoldi A, Cocorullo M, Roversi M, Chiarelli LR, Tomaiuolo M, Delre P, Mangiatordi GF, Griego A, Rizzello L, Cassetta A, Covaceuszach S, Villa S, Meneghetti F. Mori M, et al. Among authors: chiarelli lr. Pharmaceutics. 2023 Feb 2;15(2):502. doi: 10.3390/pharmaceutics15020502. Pharmaceutics. 2023. PMID: 36839823 Free PMC article.
A New Benzothiazolthiazolidine Derivative, 11726172, Is Active In Vitro, In Vivo, and against Nonreplicating Cells of Mycobacterium tuberculosis.
Salina EG, Postiglione U, Chiarelli LR, Recchia D, Záhorszká M, Lepioshkin A, Monakhova N, Pál A, Porta A, Zanoni G, Korduláková J, Kazakova E, Sassera D, Pasca MR, Makarov V, Degiacomi G. Salina EG, et al. Among authors: chiarelli lr. mSphere. 2022 Dec 21;7(6):e0036922. doi: 10.1128/msphere.00369-22. Epub 2022 Nov 15. mSphere. 2022. PMID: 36377880 Free PMC article.
Biological and structural characterization of the Mycobacterium smegmatis nitroreductase NfnB, and its role in benzothiazinone resistance.
Manina G, Bellinzoni M, Pasca MR, Neres J, Milano A, Ribeiro AL, Buroni S, Skovierová H, Dianišková P, Mikušová K, Marák J, Makarov V, Giganti D, Haouz A, Lucarelli AP, Degiacomi G, Piazza A, Chiarelli LR, De Rossi E, Salina E, Cole ST, Alzari PM, Riccardi G. Manina G, et al. Among authors: chiarelli lr. Mol Microbiol. 2010 Sep;77(5):1172-85. doi: 10.1111/j.1365-2958.2010.07277.x. Mol Microbiol. 2010. PMID: 20624223 Free article.
Analogous mechanisms of resistance to benzothiazinones and dinitrobenzamides in Mycobacterium smegmatis.
Ribeiro AL, Degiacomi G, Ewann F, Buroni S, Incandela ML, Chiarelli LR, Mori G, Kim J, Contreras-Dominguez M, Park YS, Han SJ, Brodin P, Valentini G, Rizzi M, Riccardi G, Pasca MR. Ribeiro AL, et al. Among authors: chiarelli lr. PLoS One. 2011;6(11):e26675. doi: 10.1371/journal.pone.0026675. Epub 2011 Nov 1. PLoS One. 2011. PMID: 22069462 Free PMC article.
Rv2466c mediates the activation of TP053 to kill replicating and non-replicating Mycobacterium tuberculosis.
Albesa-Jové D, Chiarelli LR, Makarov V, Pasca MR, Urresti S, Mori G, Salina E, Vocat A, Comino N, Mohorko E, Ryabova S, Pfieiffer B, Lopes Ribeiro AL, Rodrigo-Unzueta A, Tersa M, Zanoni G, Buroni S, Altmann KH, Hartkoorn RC, Glockshuber R, Cole ST, Riccardi G, Guerin ME. Albesa-Jové D, et al. Among authors: chiarelli lr. ACS Chem Biol. 2014 Jul 18;9(7):1567-75. doi: 10.1021/cb500149m. Epub 2014 Jun 13. ACS Chem Biol. 2014. PMID: 24877756 Free article.
97 results