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Optimization of Potent and Selective Ataxia Telangiectasia-Mutated Inhibitors Suitable for a Proof-of-Concept Study in Huntington's Disease Models.
J Med Chem. 2019 Mar 28;62(6):2988-3008. doi: 10.1021/acs.jmedchem.8b01819. Epub 2019 Mar 19.
J Med Chem. 2019.
PMID: 30840447
Structure-Based Exploration of Selectivity for ATM Inhibitors in Huntington's Disease.
Van de Poël A, Toledo-Sherman L, Breccia P, Cachope R, Bate JR, Angulo-Herrera I, Wishart G, Matthews KL, Martin SL, Peacock M, Barnard A, Cox HC, Jones G, McAllister G, Vater H, Esmieu W, Clissold C, Lamers M, Leonard P, Jarvis RE, Blackaby W, Eznarriaga M, Lazari O, Yates D, Rose M, Jang SW, Muñoz-Sanjuan I, Dominguez C.
Van de Poël A, et al. Among authors: angulo herrera i.
J Med Chem. 2021 Apr 22;64(8):5018-5036. doi: 10.1021/acs.jmedchem.1c00114. Epub 2021 Mar 30.
J Med Chem. 2021.
PMID: 33783225
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A novel combination treatment for fragile X syndrome predicted using computational methods.
Chadwick W, Angulo-Herrera I, Cogram P, Deacon RJM, Mason DJ, Brown D, Roberts I, O'Donovan DJ, Tranfaglia MR, Guilliams T, Thompson NT.
Chadwick W, et al. Among authors: angulo herrera i.
Brain Commun. 2024 Jan 15;6(1):fcad353. doi: 10.1093/braincomms/fcad353. eCollection 2024.
Brain Commun. 2024.
PMID: 38226317
Free PMC article.
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