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Direct activation of PP2A for the treatment of tyrosine kinase inhibitor-resistant lung adenocarcinoma.
JCI Insight. 2019 Feb 21;4(4):e125693. doi: 10.1172/jci.insight.125693. eCollection 2019 Feb 21.
JCI Insight. 2019.
PMID: 30830869
Free PMC article.
Activation of tumor suppressor protein PP2A inhibits KRAS-driven tumor growth.
Sangodkar J, Perl A, Tohme R, Kiselar J, Kastrinsky DB, Zaware N, Izadmehr S, Mazhar S, Wiredja DD, O'Connor CM, Hoon D, Dhawan NS, Schlatzer D, Yao S, Leonard D, Borczuk AC, Gokulrangan G, Wang L, Svenson E, Farrington CC, Yuan E, Avelar RA, Stachnik A, Smith B, Gidwani V, Giannini HM, McQuaid D, McClinch K, Wang Z, Levine AC, Sears RC, Chen EY, Duan Q, Datt M, Haider S, Ma'ayan A, DiFeo A, Sharma N, Galsky MD, Brautigan DL, Ioannou YA, Xu W, Chance MR, Ohlmeyer M, Narla G.
Sangodkar J, et al. Among authors: dhawan ns.
J Clin Invest. 2017 Jun 1;127(6):2081-2090. doi: 10.1172/JCI89548. Epub 2017 May 15.
J Clin Invest. 2017.
PMID: 28504649
Free PMC article.
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Targeting the FOXO1/KLF6 axis regulates EGFR signaling and treatment response.
Sangodkar J, Dhawan NS, Melville H, Singh VJ, Yuan E, Rana H, Izadmehr S, Farrington C, Mazhar S, Katz S, Albano T, Arnovitz P, Okrent R, Ohlmeyer M, Galsky M, Burstein D, Zhang D, Politi K, Difeo A, Narla G.
Sangodkar J, et al. Among authors: dhawan ns.
J Clin Invest. 2012 Jul;122(7):2637-51. doi: 10.1172/JCI62058. Epub 2012 Jun 1.
J Clin Invest. 2012.
PMID: 22653055
Free PMC article.
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Reengineered tricyclic anti-cancer agents.
Kastrinsky DB, Sangodkar J, Zaware N, Izadmehr S, Dhawan NS, Narla G, Ohlmeyer M.
Kastrinsky DB, et al. Among authors: dhawan ns.
Bioorg Med Chem. 2015 Oct 1;23(19):6528-34. doi: 10.1016/j.bmc.2015.07.007. Epub 2015 Sep 11.
Bioorg Med Chem. 2015.
PMID: 26372073
Free PMC article.
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Corrigendum to "Reengineered tricyclic anti-cancer agents" [Bioorg. Med. Chem. 23 (2015) 6528-6534].
Kastrinsky DB, Sangodkar J, Zaware N, McClinch K, Farrington CC, Giannini HM, Izadmehr S, Dhawan NS, Narla G, Ohlmeyer M.
Kastrinsky DB, et al. Among authors: dhawan ns.
Bioorg Med Chem. 2015 Dec 1;23(23):7487. doi: 10.1016/j.bmc.2015.11.002. Epub 2015 Nov 9.
Bioorg Med Chem. 2015.
PMID: 28290285
No abstract available.
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Small molecule stabilization of the KSR inactive state antagonizes oncogenic Ras signalling.
Dhawan NS, Scopton AP, Dar AC.
Dhawan NS, et al.
Nature. 2016 Sep 1;537(7618):112-116. doi: 10.1038/nature19327. Epub 2016 Aug 24.
Nature. 2016.
PMID: 27556948
Free PMC article.
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Gene-protein correlation in single cells.
Renfrow JJ, Scheck AC, Dhawan NS, Lukac PJ, Vogel H, Chandler JP, Raizer JJ, Harsh GR, Chakravarti A, Bredel M.
Renfrow JJ, et al. Among authors: dhawan ns.
Neuro Oncol. 2011 Aug;13(8):880-5. doi: 10.1093/neuonc/nor071.
Neuro Oncol. 2011.
PMID: 21798849
Free PMC article.
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