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Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity.
Botros SS, William S, Sabra AA, El-Lakkany NM, Seif El-Din SH, García-Rubia A, Sebastián-Pérez V, Blaazer AR, de Heuvel E, Sijm M, Zheng Y, Salado IG, Munday JC, Maes L, de Esch IJP, Sterk GJ, Augustyns K, Leurs R, Gil C, De Koning HP. Botros SS, et al. Among authors: augustyns k. Int J Parasitol Drugs Drug Resist. 2019 Apr;9:35-43. doi: 10.1016/j.ijpddr.2019.01.001. Epub 2019 Jan 14. Int J Parasitol Drugs Drug Resist. 2019. PMID: 30669086 Free PMC article.
Design and evaluation of Trypanosoma brucei metacaspase inhibitors.
Berg M, Van der Veken P, Joossens J, Muthusamy V, Breugelmans M, Moss CX, Rudolf J, Cos P, Coombs GH, Maes L, Haemers A, Mottram JC, Augustyns K. Berg M, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2010 Mar 15;20(6):2001-6. doi: 10.1016/j.bmcl.2010.01.099. Epub 2010 Jan 25. Bioorg Med Chem Lett. 2010. PMID: 20167486 Free PMC article.
Evaluation of nucleoside hydrolase inhibitors for treatment of African trypanosomiasis.
Berg M, Kohl L, Van der Veken P, Joossens J, Al-Salabi MI, Castagna V, Giannese F, Cos P, Versées W, Steyaert J, Grellier P, Haemers A, Degano M, Maes L, de Koning HP, Augustyns K. Berg M, et al. Among authors: augustyns k. Antimicrob Agents Chemother. 2010 May;54(5):1900-8. doi: 10.1128/AAC.01787-09. Epub 2010 Mar 1. Antimicrob Agents Chemother. 2010. PMID: 20194690 Free PMC article.
α-ketoheterocycles as inhibitors of Leishmania mexicana cysteine protease CPB.
Steert K, Berg M, Mottram JC, Westrop GD, Coombs GH, Cos P, Maes L, Joossens J, Van der Veken P, Haemers A, Augustyns K. Steert K, et al. Among authors: augustyns k. ChemMedChem. 2010 Oct 4;5(10):1734-48. doi: 10.1002/cmdc.201000265. ChemMedChem. 2010. PMID: 20799311 Free PMC article.
Novel triazine dimers with potent antitrypanosomal activity.
Venkatraj M, Salado IG, Heeres J, Joossens J, Lewi PJ, Caljon G, Maes L, Van der Veken P, Augustyns K. Venkatraj M, et al. Among authors: augustyns k. Eur J Med Chem. 2018 Jan 1;143:306-319. doi: 10.1016/j.ejmech.2017.11.075. Epub 2017 Nov 27. Eur J Med Chem. 2018. PMID: 29197735
α-Amino Diphenyl Phosphonates as Novel Inhibitors of Escherichia coli ClpP Protease.
Moreno-Cinos C, Sassetti E, Salado IG, Witt G, Benramdane S, Reinhardt L, Cruz CD, Joossens J, Van der Veken P, Brötz-Oesterhelt H, Tammela P, Winterhalter M, Gribbon P, Windshügel B, Augustyns K. Moreno-Cinos C, et al. Among authors: augustyns k. J Med Chem. 2019 Jan 24;62(2):774-797. doi: 10.1021/acs.jmedchem.8b01466. Epub 2019 Jan 11. J Med Chem. 2019. PMID: 30571121
ClpP Protease, a Promising Antimicrobial Target.
Moreno-Cinos C, Goossens K, Salado IG, Van Der Veken P, De Winter H, Augustyns K. Moreno-Cinos C, et al. Among authors: augustyns k. Int J Mol Sci. 2019 May 7;20(9):2232. doi: 10.3390/ijms20092232. Int J Mol Sci. 2019. PMID: 31067645 Free PMC article. Review.
Evaluation of phthalazinone phosphodiesterase inhibitors with improved activity and selectivity against Trypanosoma cruzi.
De Araújo JS, da Silva PB, Batista MM, Peres RB, Cardoso-Santos C, Kalejaiye TD, Munday JC, De Heuvel E, Sterk GJ, Augustyns K, Salado IG, Matheeussen A, De Esch I, De Koning HP, Leurs R, Maes L, Soeiro MNC. De Araújo JS, et al. Among authors: augustyns k. J Antimicrob Chemother. 2020 Apr 1;75(4):958-967. doi: 10.1093/jac/dkz516. J Antimicrob Chemother. 2020. PMID: 31860098
175 results