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The MAP kinase-interacting kinases (MNKs) as targets in oncology.
Expert Opin Ther Targets. 2019 Mar;23(3):187-199. doi: 10.1080/14728222.2019.1571043. Epub 2019 Jan 24.
Expert Opin Ther Targets. 2019.
PMID: 30650992
Review.
Reciprocal signaling between mTORC1 and MNK2 controls cell growth and oncogenesis.
Xie J, Shen K, Jones AT, Yang J, Tee AR, Shen MH, Yu M, Irani S, Wong D, Merrett JE, Lenchine RV, De Poi S, Jensen KB, Trim PJ, Snel MF, Kamei M, Martin SK, Fitter S, Tian S, Wang X, Butler LM, Zannettino ACW, Proud CG.
Xie J, et al. Among authors: merrett je.
Cell Mol Life Sci. 2021 Jan;78(1):249-270. doi: 10.1007/s00018-020-03491-1. Epub 2020 Mar 13.
Cell Mol Life Sci. 2021.
PMID: 32170339
Free PMC article.
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MAPK-interacting kinase 2 (MNK2) regulates adipocyte metabolism independently of its catalytic activity.
Merrett JE, Xie J, Psaltis PJ, Proud CG.
Merrett JE, et al.
Biochem J. 2020 Jul 31;477(14):2735-2754. doi: 10.1042/BCJ20200433.
Biochem J. 2020.
PMID: 32648926
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Design, synthesis and activity of Mnk1 and Mnk2 selective inhibitors containing thieno[2,3-d]pyrimidine scaffold.
Jin X, Merrett J, Tong S, Flower B, Xie J, Yu R, Tian S, Gao L, Zhao J, Wang X, Jiang T, Proud CG.
Jin X, et al.
Eur J Med Chem. 2019 Jan 15;162:735-751. doi: 10.1016/j.ejmech.2018.10.070. Epub 2018 Nov 2.
Eur J Med Chem. 2019.
PMID: 30496989
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Identification of DNA response elements regulating expression of CCAAT/enhancer-binding protein (C/EBP) β and δ and MAP kinase-interacting kinases during early adipogenesis.
Merrett JE, Bo T, Psaltis PJ, Proud CG.
Merrett JE, et al.
Adipocyte. 2020 Dec;9(1):427-442. doi: 10.1080/21623945.2020.1796361.
Adipocyte. 2020.
PMID: 32787498
Free PMC article.
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