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Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR.
Annunziato G, Pieroni M, Benoni R, Campanini B, Pertinhez TA, Pecchini C, Bruno A, Magalhães J, Bettati S, Franko N, Mozzarelli A, Costantino G. Annunziato G, et al. J Enzyme Inhib Med Chem. 2016;31(sup4):78-87. doi: 10.1080/14756366.2016.1218486. Epub 2016 Aug 31. J Enzyme Inhib Med Chem. 2016. PMID: 27578398
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents.
Pieroni M, Azzali E, Basilico N, Parapini S, Zolkiewski M, Beato C, Annunziato G, Bruno A, Vacondio F, Costantino G. Pieroni M, et al. Among authors: annunziato g. J Med Chem. 2017 Mar 9;60(5):1959-1970. doi: 10.1021/acs.jmedchem.6b01685. Epub 2017 Feb 14. J Med Chem. 2017. PMID: 28128956
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug design.
Magalhães J, Franko N, Annunziato G, Welch M, Dolan SK, Bruno A, Mozzarelli A, Armao S, Jirgensons A, Pieroni M, Costantino G, Campanini B. Magalhães J, et al. Among authors: annunziato g. J Enzyme Inhib Med Chem. 2018 Dec;33(1):1444-1452. doi: 10.1080/14756366.2018.1512596. J Enzyme Inhib Med Chem. 2018. PMID: 30221554 Free PMC article.
Refining the structure-activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms.
Magalhães J, Franko N, Annunziato G, Pieroni M, Benoni R, Nikitjuka A, Mozzarelli A, Bettati S, Karawajczyk A, Jirgensons A, Campanini B, Costantino G. Magalhães J, et al. Among authors: annunziato g. J Enzyme Inhib Med Chem. 2019 Dec;34(1):31-43. doi: 10.1080/14756366.2018.1518959. J Enzyme Inhib Med Chem. 2019. PMID: 30362368 Free PMC article.
24 results