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Easy-To-Synthesize Spirocyclic Compounds Possess Remarkable in Vivo Activity against Mycobacterium tuberculosis.
J Med Chem. 2018 Dec 27;61(24):11327-11340. doi: 10.1021/acs.jmedchem.8b01533. Epub 2018 Dec 12.
J Med Chem. 2018.
PMID: 30457865
Inhibitory Kappa B Kinase α (IKKα) Inhibitors That Recapitulate Their Selectivity in Cells against Isoform-Related Biomarkers.
Anthony NG, Baiget J, Berretta G, Boyd M, Breen D, Edwards J, Gamble C, Gray AI, Harvey AL, Hatziieremia S, Ho KH, Huggan JK, Lang S, Llona-Minguez S, Luo JL, McIntosh K, Paul A, Plevin RJ, Robertson MN, Scott R, Suckling CJ, Sutcliffe OB, Young LC, Mackay SP.
Anthony NG, et al. Among authors: baiget j.
J Med Chem. 2017 Aug 24;60(16):7043-7066. doi: 10.1021/acs.jmedchem.7b00484. Epub 2017 Aug 15.
J Med Chem. 2017.
PMID: 28737909
Free PMC article.
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Topographical Mapping of Isoform-Selectivity Determinants for J-Channel-Binding Inhibitors of Sphingosine Kinases 1 and 2.
Adams DR, Tawati S, Berretta G, Rivas PL, Baiget J, Jiang Z, Alsfouk A, Mackay SP, Pyne NJ, Pyne S.
Adams DR, et al. Among authors: baiget j.
J Med Chem. 2019 Apr 11;62(7):3658-3676. doi: 10.1021/acs.jmedchem.9b00162. Epub 2019 Mar 27.
J Med Chem. 2019.
PMID: 30889352
Free article.
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Manganese dioxide mediated one-pot synthesis of methyl 9H-pyrido[3,4-b]indole-1-carboxylate: Concise synthesis of alangiobussinine.
Baiget J, Llona-Minguez S, Lang S, Mackay SP, Suckling CJ, Sutcliffe OB.
Baiget J, et al.
Beilstein J Org Chem. 2011;7:1407-11. doi: 10.3762/bjoc.7.164. Epub 2011 Oct 12.
Beilstein J Org Chem. 2011.
PMID: 22043251
Free PMC article.
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Small-molecule inhibitors of IκB kinase (IKK) and IKK-related kinases.
Llona-Minguez S, Baiget J, Mackay SP.
Llona-Minguez S, et al. Among authors: baiget j.
Pharm Pat Anal. 2013 Jul;2(4):481-98. doi: 10.4155/ppa.13.31.
Pharm Pat Anal. 2013.
PMID: 24237125
Review.
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Diastereoselective additions of titanium enolates from N-glycolyl thiazolidinethiones to acetals.
Baiget J, Caba M, Gálvez E, Romea P, Urpí F, Font-Bardia M.
Baiget J, et al.
J Org Chem. 2012 Oct 5;77(19):8809-14. doi: 10.1021/jo301569x. Epub 2012 Sep 18.
J Org Chem. 2012.
PMID: 22985246
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