Giannini G - Search Results

1

Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation.

Cini E, Faltoni V, Petricci E, Taddei M, Salvini L, Giannini G, Vesci L, Milazzo FM, Anastasi AM, Battistuzzi G, De Santis R. Cini E, et al. Among authors: giannini g. Chem Sci. 2018 Jul 3;9(31):6490-6496. doi: 10.1039/c7sc05266a. eCollection 2018 Aug 21. Chem Sci. 2018. PMID: 30288233 Free PMC article.

2

E-ring-modified 7-oxyiminomethyl camptothecins: Synthesis and preliminary in vitro and in vivo biological evaluation.

Giannini G, Marzi M, Cabri W, Marastoni E, Battistuzzi G, Vesci L, Pisano C, Beretta GL, De Cesare M, Zunino F. Giannini G, et al. Bioorg Med Chem Lett. 2008 May 1;18(9):2910-5. doi: 10.1016/j.bmcl.2008.03.074. Epub 2008 Mar 30. Bioorg Med Chem Lett. 2008. PMID: 18424133

3

N-Hydroxy-(4-oxime)-cinnamide: a versatile scaffold for the synthesis of novel histone deacetylase [correction of deacetilase] (HDAC) inhibitors.

Giannini G, Marzi M, Pezzi R, Brunetti T, Battistuzzi G, Marzo MD, Cabri W, Vesci L, Pisano C. Giannini G, et al. Bioorg Med Chem Lett. 2009 Apr 15;19(8):2346-9. doi: 10.1016/j.bmcl.2009.02.029. Epub 2009 Feb 12. Bioorg Med Chem Lett. 2009. PMID: 19285395

4

Exploring bis-(indolyl)methane moiety as an alternative and innovative CAP group in the design of histone deacetylase (HDAC) inhibitors.

Giannini G, Marzi M, Marzo MD, Battistuzzi G, Pezzi R, Brunetti T, Cabri W, Vesci L, Pisano C. Giannini G, et al. Bioorg Med Chem Lett. 2009 May 15;19(10):2840-3. doi: 10.1016/j.bmcl.2009.03.101. Epub 2009 Mar 26. Bioorg Med Chem Lett. 2009. PMID: 19359173

5

Novel tumor-targeted RGD peptide-camptothecin conjugates: synthesis and biological evaluation.

Dal Pozzo A, Ni MH, Esposito E, Dallavalle S, Musso L, Bargiotti A, Pisano C, Vesci L, Bucci F, Castorina M, Foderà R, Giannini G, Aulicino C, Penco S. Dal Pozzo A, et al. Among authors: giannini g. Bioorg Med Chem. 2010 Jan 1;18(1):64-72. doi: 10.1016/j.bmc.2009.11.019. Epub 2009 Nov 12. Bioorg Med Chem. 2010. PMID: 19942441

6

Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors.

Musso L, Dallavalle S, Merlini L, Bava A, Nasini G, Penco S, Giannini G, Giommarelli C, De Cesare A, Zuco V, Vesci L, Pisano C, Castorina M, Milazzo F, Cervoni ML, Dal Piaz F, De Tommasi N, Zunino F. Musso L, et al. Among authors: giannini g. Bioorg Med Chem. 2010 Aug 15;18(16):6031-43. doi: 10.1016/j.bmc.2010.06.068. Epub 2010 Jul 1. Bioorg Med Chem. 2010. PMID: 20655237

7

Non-natural macrocyclic inhibitors of histone deacetylases: design, synthesis, and activity.

Auzzas L, Larsson A, Matera R, Baraldi A, Deschênes-Simard B, Giannini G, Cabri W, Battistuzzi G, Gallo G, Ciacci A, Vesci L, Pisano C, Hanessian S. Auzzas L, et al. Among authors: giannini g. J Med Chem. 2010 Dec 9;53(23):8387-99. doi: 10.1021/jm101092u. Epub 2010 Nov 12. J Med Chem. 2010. PMID: 21073160

8

Oxime amides as a novel zinc binding group in histone deacetylase inhibitors: synthesis, biological activity, and computational evaluation.

Botta CB, Cabri W, Cini E, De Cesare L, Fattorusso C, Giannini G, Persico M, Petrella A, Rondinelli F, Rodriquez M, Russo A, Taddei M. Botta CB, et al. Among authors: giannini g. J Med Chem. 2011 Apr 14;54(7):2165-82. doi: 10.1021/jm101373a. Epub 2011 Mar 18. J Med Chem. 2011. PMID: 21417297

9

Novel 3,4-isoxazolediamides as potent inhibitors of chaperone heat shock protein 90.

Baruchello R, Simoni D, Grisolia G, Barbato G, Marchetti P, Rondanin R, Mangiola S, Giannini G, Brunetti T, Alloatti D, Gallo G, Ciacci A, Vesci L, Castorina M, Milazzo FM, Cervoni ML, Guglielmi MB, Barbarino M, Foderà R, Pisano C, Cabri W. Baruchello R, et al. Among authors: giannini g. J Med Chem. 2011 Dec 22;54(24):8592-604. doi: 10.1021/jm201155e. Epub 2011 Nov 23. J Med Chem. 2011. PMID: 22066525

10

New retinoid derivatives as back-ups of Adarotene.

Giannini G, Brunetti T, Battistuzzi G, Alloatti D, Quattrociocchi G, Cima MG, Merlini L, Dallavalle S, Cincinelli R, Nannei R, Vesci L, Bucci F, Foderà R, Guglielmi MB, Pisano C, Cabri W. Giannini G, et al. Bioorg Med Chem. 2012 Apr 1;20(7):2405-15. doi: 10.1016/j.bmc.2012.01.042. Epub 2012 Feb 6. Bioorg Med Chem. 2012. PMID: 22365912

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