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Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation.
Chem Sci. 2018 Jul 3;9(31):6490-6496. doi: 10.1039/c7sc05266a. eCollection 2018 Aug 21.
Chem Sci. 2018.
PMID: 30288233
Free PMC article.
Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition.
Cianferotti C, Faltoni V, Cini E, Ermini E, Migliorini F, Petricci E, Taddei M, Salvini L, Battistuzzi G, Milazzo FM, Anastasi AM, Chiapparino C, De Santis R, Giannini G.
Cianferotti C, et al. Among authors: faltoni v.
Chem Commun (Camb). 2021 Jan 28;57(7):867-870. doi: 10.1039/d0cc06131j.
Chem Commun (Camb). 2021.
PMID: 33433550
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ErbB2 Targeted Epigenetic Modulation: Anti-tumor Efficacy of the ADC Trastuzumab-HDACi ST8176AA1.
Milazzo FM, Vesci L, Anastasi AM, Chiapparino C, Rosi A, Giannini G, Taddei M, Cini E, Faltoni V, Petricci E, Battistuzzi G, Salvini L, Carollo V, De Santis R.
Milazzo FM, et al. Among authors: faltoni v.
Front Oncol. 2020 Jan 23;9:1534. doi: 10.3389/fonc.2019.01534. eCollection 2019.
Front Oncol. 2020.
PMID: 32039017
Free PMC article.
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