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Structure-activity relationship study on anti-HIV 6-desfluoroquinolones.
Tabarrini O, Massari S, Daelemans D, Stevens M, Manfroni G, Sabatini S, Balzarini J, Cecchetti V, Pannecouque C, Fravolini A. Tabarrini O, et al. J Med Chem. 2008 Sep 11;51(17):5454-8. doi: 10.1021/jm701585h. Epub 2008 Aug 19. J Med Chem. 2008. PMID: 18710207
Studies on anti-HIV quinolones: new insights on the C-6 position.
Massari S, Daelemans D, Manfroni G, Sabatini S, Tabarrini O, Pannecouque C, Cecchetti V. Massari S, et al. Among authors: tabarrini o. Bioorg Med Chem. 2009 Jan 15;17(2):667-74. doi: 10.1016/j.bmc.2008.11.056. Epub 2008 Dec 3. Bioorg Med Chem. 2009. PMID: 19091580
2-Phenylquinolones as inhibitors of the HIV-1 Tat-TAR interaction.
Gatto B, Tabarrini O, Massari S, Giaretta G, Sabatini S, Del Vecchio C, Parolin C, Fravolini A, Palumbo M, Cecchetti V. Gatto B, et al. Among authors: tabarrini o. ChemMedChem. 2009 Jun;4(6):935-8. doi: 10.1002/cmdc.200800437. ChemMedChem. 2009. PMID: 19283692
118 results