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Structure-based design and profiling of novel 17β-HSD14 inhibitors.
Braun F, Bertoletti N, Möller G, Adamski J, Frotscher M, Guragossian N, Madeira Gírio PA, Le Borgne M, Ettouati L, Falson P, Müller S, Vollmer G, Heine A, Klebe G, Marchais-Oberwinkler S. Braun F, et al. Among authors: bertoletti n. Eur J Med Chem. 2018 Jul 15;155:61-76. doi: 10.1016/j.ejmech.2018.05.029. Epub 2018 May 22. Eur J Med Chem. 2018. PMID: 29859505
First Structure-Activity Relationship of 17β-Hydroxysteroid Dehydrogenase Type 14 Nonsteroidal Inhibitors and Crystal Structures in Complex with the Enzyme.
Braun F, Bertoletti N, Möller G, Adamski J, Steinmetzer T, Salah M, Abdelsamie AS, van Koppen CJ, Heine A, Klebe G, Marchais-Oberwinkler S. Braun F, et al. Among authors: bertoletti n. J Med Chem. 2016 Dec 8;59(23):10719-10737. doi: 10.1021/acs.jmedchem.6b01436. Epub 2016 Nov 18. J Med Chem. 2016. PMID: 27933965
Structure-Guided Identification of DNMT3B Inhibitors.
Newton AS, Faver JC, Micevic G, Muthusamy V, Kudalkar SN, Bertoletti N, Anderson KS, Bosenberg MW, Jorgensen WL. Newton AS, et al. Among authors: bertoletti n. ACS Med Chem Lett. 2020 Feb 7;11(5):971-976. doi: 10.1021/acsmedchemlett.0c00011. eCollection 2020 May 14. ACS Med Chem Lett. 2020. PMID: 32435413 Free PMC article.
Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV.
Kudalkar SN, Ullah I, Bertoletti N, Mandl HK, Cisneros JA, Beloor J, Chan AH, Quijano E, Saltzman WM, Jorgensen WL, Kumar P, Anderson KS. Kudalkar SN, et al. Among authors: bertoletti n. Antiviral Res. 2019 Jul;167:110-116. doi: 10.1016/j.antiviral.2019.04.010. Epub 2019 Apr 26. Antiviral Res. 2019. PMID: 31034849 Free PMC article.
Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead.
Ippolito JA, Niu H, Bertoletti N, Carter ZJ, Jin S, Spasov KA, Cisneros JA, Valhondo M, Cutrona KJ, Anderson KS, Jorgensen WL. Ippolito JA, et al. Among authors: bertoletti n. ACS Med Chem Lett. 2021 Jan 6;12(2):249-255. doi: 10.1021/acsmedchemlett.0c00612. eCollection 2021 Feb 11. ACS Med Chem Lett. 2021. PMID: 33603971 Free PMC article.
Structural Studies and Structure Activity Relationships for Novel Computationally Designed Non-nucleoside Inhibitors and Their Interactions With HIV-1 Reverse Transcriptase.
Frey KM, Bertoletti N, Chan AH, Ippolito JA, Bollini M, Spasov KA, Jorgensen WL, Anderson KS. Frey KM, et al. Among authors: bertoletti n. Front Mol Biosci. 2022 Feb 14;9:805187. doi: 10.3389/fmolb.2022.805187. eCollection 2022. Front Mol Biosci. 2022. PMID: 35237658 Free PMC article.
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