Gratteri P - Search Results

1

Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform.

Ibrahim HS, Allam HA, Mahmoud WR, Bonardi A, Nocentini A, Gratteri P, Ibrahim ES, Abdel-Aziz HA, Supuran CT. Ibrahim HS, et al. Among authors: gratteri p. Eur J Med Chem. 2018 May 25;152:1-9. doi: 10.1016/j.ejmech.2018.04.016. Epub 2018 Apr 10. Eur J Med Chem. 2018. PMID: 29684705

2

Synthesis and benzodiazepine receptor affinity of pyrazolo[1,5-a]pyrimidine derivatives. 3. New 6-(3-thienyl) series as alpha 1 selective ligands.

Selleri S, Bruni F, Costagli C, Costanzo A, Guerrini G, Ciciani G, Gratteri P, Bonaccini C, Malmberg Aiello P, Besnard F, Renard S, Costa B, Martini C. Selleri S, et al. Among authors: gratteri p. J Med Chem. 2003 Jan 16;46(2):310-3. doi: 10.1021/jm020999w. J Med Chem. 2003. PMID: 12519068

3

Field interaction and geometrical overlap: a new simplex and experimental design based computational procedure for superposing small ligand molecules.

Melani F, Gratteri P, Adamo M, Bonaccini C. Melani F, et al. Among authors: gratteri p. J Med Chem. 2003 Apr 10;46(8):1359-71. doi: 10.1021/jm0210616. J Med Chem. 2003. PMID: 12672236

4

Searching for a reliable orientation of ligands in their binding site: comparison between a structure-based (Glide) and a ligand-based (FIGO) approach in the case study of PDE4 inhibitors.

Gratteri P, Bonaccini C, Melani F. Gratteri P, et al. J Med Chem. 2005 Mar 10;48(5):1657-65. doi: 10.1021/jm049289b. J Med Chem. 2005. PMID: 15743207

5

Insight into 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamides as peripheral benzodiazepine receptor ligands: synthesis, biological evaluation and 3D-QSAR investigation.

Selleri S, Gratteri P, Costagli C, Bonaccini C, Costanzo A, Melani F, Guerrini G, Ciciani G, Costa B, Spinetti F, Martini C, Bruni F. Selleri S, et al. Among authors: gratteri p. Bioorg Med Chem. 2005 Aug 15;13(16):4821-34. doi: 10.1016/j.bmc.2005.05.015. Bioorg Med Chem. 2005. PMID: 15975799

6

A novel selective GABA(A) alpha1 receptor agonist displaying sedative and anxiolytic-like properties in rodents.

Selleri S, Bruni F, Costagli C, Costanzo A, Guerrini G, Ciciani G, Gratteri P, Besnard F, Costa B, Montali M, Martini C, Fohlin J, De Siena G, Aiello PM. Selleri S, et al. Among authors: gratteri p. J Med Chem. 2005 Oct 20;48(21):6756-60. doi: 10.1021/jm058002n. J Med Chem. 2005. PMID: 16220991

7

Structural investigation of the 7-chloro-3-hydroxy-1H-quinazoline-2,4-dione scaffold to obtain AMPA and kainate receptor selective antagonists. Synthesis, pharmacological, and molecular modeling studies.

Colotta V, Catarzi D, Varano F, Lenzi O, Filacchioni G, Costagli C, Galli A, Ghelardini C, Galeotti N, Gratteri P, Sgrignani J, Deflorian F, Moro S. Colotta V, et al. Among authors: gratteri p. J Med Chem. 2006 Oct 5;49(20):6015-26. doi: 10.1021/jm0604880. J Med Chem. 2006. PMID: 17004715

8

Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin alphavbeta3 and alphavbeta5 ligands.

Salvati M, Cordero FM, Pisaneschi F, Melani F, Gratteri P, Cini N, Bottoncetti A, Brandi A. Salvati M, et al. Among authors: gratteri p. Bioorg Med Chem. 2008 Apr 15;16(8):4262-71. doi: 10.1016/j.bmc.2008.02.080. Epub 2008 Feb 29. Bioorg Med Chem. 2008. PMID: 18343671

9

Solution and Solid-State Analysis of Binding of 13-Substituted Berberine Analogues to Human Telomeric G-quadruplexes.

Ferraroni M, Bazzicalupi C, Papi F, Fiorillo G, Guamán-Ortiz LM, Nocentini A, Scovassi AI, Lombardi P, Gratteri P. Ferraroni M, et al. Among authors: gratteri p. Chem Asian J. 2016 Apr 5;11(7):1107-15. doi: 10.1002/asia.201600116. Epub 2016 Mar 11. Chem Asian J. 2016. PMID: 26865223

10

Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations.

Nocentini A, Ferraroni M, Carta F, Ceruso M, Gratteri P, Lanzi C, Masini E, Supuran CT. Nocentini A, et al. Among authors: gratteri p. J Med Chem. 2016 Dec 8;59(23):10692-10704. doi: 10.1021/acs.jmedchem.6b01389. Epub 2016 Nov 21. J Med Chem. 2016. PMID: 27933963

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

139 results

Search Page