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2-Aminoquinazolin-4(3H)-one based plasmepsin inhibitors with improved hydrophilicity and selectivity.
Bioorg Med Chem. 2018 May 15;26(9):2488-2500. doi: 10.1016/j.bmc.2018.04.012. Epub 2018 Apr 5.
Bioorg Med Chem. 2018.
PMID: 29636223
Fragment-Based Discovery of 2-Aminoquinazolin-4(3H)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV.
Rasina D, Otikovs M, Leitans J, Recacha R, Borysov OV, Kanepe-Lapsa I, Domraceva I, Pantelejevs T, Tars K, Blackman MJ, Jaudzems K, Jirgensons A.
Rasina D, et al. Among authors: borysov ov.
J Med Chem. 2016 Jan 14;59(1):374-87. doi: 10.1021/acs.jmedchem.5b01558. Epub 2015 Dec 23.
J Med Chem. 2016.
PMID: 26670264
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Synthesis of 5-(Fluoroalkyl)isoxazole Building Blocks by Regioselective Reactions of Functionalized Halogenoximes.
Chalyk BA, Hrebeniuk KV, Fil YV, Gavrilenko KS, Rozhenko AB, Vashchenko BV, Borysov OV, Biitseva AV, Lebed PS, Bakanovych I, Moroz YS, Grygorenko OO.
Chalyk BA, et al. Among authors: borysov ov.
J Org Chem. 2019 Dec 20;84(24):15877-15899. doi: 10.1021/acs.joc.9b02264. Epub 2019 Oct 30.
J Org Chem. 2019.
PMID: 31626546
Free PMC article.
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Spiropyran-Based Photoisomerizable α-Amino Acid for Membrane-Active Peptide Modification.
Hrebonkin A, Afonin S, Nikitjuka A, Borysov OV, Leitis G, Babii O, Koniev S, Lorig T, Grage SL, Nick P, Ulrich AS, Jirgensons A, Komarov IV.
Hrebonkin A, et al. Among authors: borysov ov.
Chemistry. 2024 Apr 16;30(22):e202400066. doi: 10.1002/chem.202400066. Epub 2024 Mar 1.
Chemistry. 2024.
PMID: 38366887
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Synthesis of methotrexate-betulonic acid hybrids and evaluation of their effect on artificial and Caco-2 cell membranes.
Semenenko OM, Lipson VV, Sadchenko AO, Vashchenko OV, Kasian NA, Sviechnikova LV, Lisetski LM, Babak ML, Vakula VM, Borysov OV, Holota YV, Zozulya SO, Borysko PO, Mazepa OV.
Semenenko OM, et al. Among authors: borysov ov.
Steroids. 2024 Jan;201:109332. doi: 10.1016/j.steroids.2023.109332. Epub 2023 Nov 7.
Steroids. 2024.
PMID: 37939980
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