Affron DP - Search Results

1

High-Throughput Kinetic Analysis for Target-Directed Covalent Ligand Discovery.

Craven GB, Affron DP, Allen CE, Matthies S, Greener JG, Morgan RML, Tate EW, Armstrong A, Mann DJ. Craven GB, et al. Among authors: affron dp. Angew Chem Int Ed Engl. 2018 May 4;57(19):5257-5261. doi: 10.1002/anie.201711825. Epub 2018 Mar 26. Angew Chem Int Ed Engl. 2018. PMID: 29480525 Free PMC article.

2

Multiparameter Kinetic Analysis for Covalent Fragment Optimization by Using Quantitative Irreversible Tethering (qIT).

Craven GB, Affron DP, Kösel T, Wong TLM, Jukes ZH, Liu CT, Morgan RML, Armstrong A, Mann DJ. Craven GB, et al. Among authors: affron dp. Chembiochem. 2020 Dec 1;21(23):3417-3422. doi: 10.1002/cbic.202000457. Epub 2020 Aug 7. Chembiochem. 2020. PMID: 32659037 Free PMC article.

3

Vinyl sulfonamide synthesis for irreversible tethering via a novel α-selenoether protection strategy.

Craven GB, Affron DP, Raymond PN, Mann DJ, Armstrong A. Craven GB, et al. Among authors: affron dp. Medchemcomm. 2018 Dec 13;10(1):158-163. doi: 10.1039/c8md00566d. eCollection 2019 Jan 1. Medchemcomm. 2018. PMID: 30774862 Free PMC article.

4

Synthesis and Configurational Assignment of Vinyl Sulfoximines and Sulfonimidamides.

Craven GB, Briggs EL, Zammit CM, McDermott A, Greed S, Affron DP, Leinfellner C, Cudmore HR, Tweedy RR, Luisi R, Bull JA, Armstrong A. Craven GB, et al. Among authors: affron dp. J Org Chem. 2021 Jun 4;86(11):7403-7424. doi: 10.1021/acs.joc.1c00373. Epub 2021 May 18. J Org Chem. 2021. PMID: 34003635

5

Rapid Assembly of Saturated Nitrogen Heterocycles in One-Pot: Diazo-Heterocycle "Stitching" by N-H Insertion and Cyclization.

Boddy AJ, Affron DP, Cordier CJ, Rivers EL, Spivey AC, Bull JA. Boddy AJ, et al. Among authors: affron dp. Angew Chem Int Ed Engl. 2019 Jan 28;58(5):1458-1462. doi: 10.1002/anie.201812925. Epub 2018 Dec 28. Angew Chem Int Ed Engl. 2019. PMID: 30516342 Free article.

6

Synthesis of cis-C-iodo-N-tosyl-aziridines using diiodomethyllithium: reaction optimization, product scope and stability, and a protocol for selection of stationary phase for chromatography.

Boultwood T, Affron DP, Trowbridge AD, Bull JA. Boultwood T, et al. Among authors: affron dp. J Org Chem. 2013 Jul 5;78(13):6632-47. doi: 10.1021/jo400956x. Epub 2013 Jun 18. J Org Chem. 2013. PMID: 23738857 Free PMC article.

7

Palladium-Catalyzed Directed C(sp³)-H Arylation of Saturated Heterocycles at C-3 Using a Concise Optimization Approach.

Affron DP, Bull JA. Affron DP, et al. European J Org Chem. 2016 Jan;2016(1):139-149. doi: 10.1002/ejoc.201501300. Epub 2015 Nov 27. European J Org Chem. 2016. PMID: 26877706 Free PMC article.

8

Regio- and stereospecific synthesis of C-3 functionalized proline derivatives by palladium catalyzed directed C(sp3)-H arylation.

Affron DP, Davis OA, Bull JA. Affron DP, et al. Org Lett. 2014 Sep 19;16(18):4956-9. doi: 10.1021/ol502511g. Epub 2014 Sep 5. Org Lett. 2014. PMID: 25191995 Free article.

9

Regio- and Stereoselective Palladium-Catalyzed C(sp³)-H Arylation of Pyrrolidines and Piperidines with C(3) Directing Groups.

Antermite D, Affron DP, Bull JA. Antermite D, et al. Among authors: affron dp. Org Lett. 2018 Jul 6;20(13):3948-3952. doi: 10.1021/acs.orglett.8b01521. Epub 2018 Jun 13. Org Lett. 2018. PMID: 29897773 Free article.

10

Synthesis and purification of iodoaziridines involving quantitative selection of the optimal stationary phase for chromatography.

Boultwood T, Affron DP, Bull JA. Boultwood T, et al. Among authors: affron dp. J Vis Exp. 2014 May 16;(87):51633. doi: 10.3791/51633. J Vis Exp. 2014. PMID: 24893769 Free PMC article.

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