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( S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation.
J Med Chem. 2018 Mar 8;61(5):2124-2130. doi: 10.1021/acs.jmedchem.8b00099. Epub 2018 Feb 26.
J Med Chem. 2018.
PMID: 29451794
A stereoselective approach to peptidomimetic BACE1 inhibitors.
Butini S, Gabellieri E, Brindisi M, Giovani S, Maramai S, Kshirsagar G, Guarino E, Brogi S, La Pietra V, Giustiniano M, Marinelli L, Novellino E, Campiani G, Cappelli A, Gemma S.
Butini S, et al.
Eur J Med Chem. 2013;70:233-47. doi: 10.1016/j.ejmech.2013.09.056. Epub 2013 Oct 6.
Eur J Med Chem. 2013.
PMID: 24158015
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Ionotropic Glutamate Receptor GluA2 in Complex with Bicyclic Pyrimidinedione-Based Compounds: When Small Compound Modifications Have Distinct Effects on Binding Interactions.
Frydenvang K, Pickering DS, Kshirsagar GU, Chemi G, Gemma S, Sprogøe D, Kærn AM, Brogi S, Campiani G, Butini S, Kastrup JS.
Frydenvang K, et al. Among authors: kshirsagar gu.
ACS Chem Neurosci. 2020 Jun 17;11(12):1791-1800. doi: 10.1021/acschemneuro.0c00195. Epub 2020 Jun 5.
ACS Chem Neurosci. 2020.
PMID: 32437601
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