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Structure-Function Evaluation of Imidazopyridine Derivatives Selective for δ-Subunit-Containing γ-Aminobutyric Acid Type A (GABAA) Receptors.
Yakoub K, Jung S, Sattler C, Damerow H, Weber J, Kretzschmann A, Cankaya AS, Piel M, Rösch F, Haugaard AS, Frølund B, Schirmeister T, Lüddens H. Yakoub K, et al. Among authors: schirmeister t. J Med Chem. 2018 Mar 8;61(5):1951-1968. doi: 10.1021/acs.jmedchem.7b01484. Epub 2018 Feb 26. J Med Chem. 2018. PMID: 29451785
Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation.
Ettari R, Pinto A, Previti S, Tamborini L, Angelo IC, La Pietra V, Marinelli L, Novellino E, Schirmeister T, Zappalà M, Grasso S, De Micheli C, Conti P. Ettari R, et al. Among authors: schirmeister t. Bioorg Med Chem. 2015 Nov 1;23(21):7053-60. doi: 10.1016/j.bmc.2015.09.029. Epub 2015 Sep 21. Bioorg Med Chem. 2015. PMID: 26432608
Bistacrine derivatives as new potent antimalarials.
Schmidt I, Pradel G, Sologub L, Golzmann A, Ngwa CJ, Kucharski A, Schirmeister T, Holzgrabe U. Schmidt I, et al. Among authors: schirmeister t. Bioorg Med Chem. 2016 Aug 15;24(16):3636-42. doi: 10.1016/j.bmc.2016.06.003. Epub 2016 Jun 4. Bioorg Med Chem. 2016. PMID: 27316542
Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure-based virtual screening.
Di Giovanni C, Ettari R, Sarno S, Rotondo A, Bitto A, Squadrito F, Altavilla D, Schirmeister T, Novellino E, Grasso S, Zappalà M, Lavecchia A. Di Giovanni C, et al. Among authors: schirmeister t. Eur J Med Chem. 2016 Oct 4;121:578-591. doi: 10.1016/j.ejmech.2016.05.049. Epub 2016 May 27. Eur J Med Chem. 2016. PMID: 27318981
Dipeptidyl Nitroalkenes as Potent Reversible Inhibitors of Cysteine Proteases Rhodesain and Cruzain.
Latorre A, Schirmeister T, Kesselring J, Jung S, Johé P, Hellmich UA, Heilos A, Engels B, Krauth-Siegel RL, Dirdjaja N, Bou-Iserte L, Rodríguez S, González FV. Latorre A, et al. Among authors: schirmeister t. ACS Med Chem Lett. 2016 Sep 21;7(12):1073-1076. doi: 10.1021/acsmedchemlett.6b00276. eCollection 2016 Dec 8. ACS Med Chem Lett. 2016. PMID: 27994740 Free PMC article.
Synthesis and Pharmacological Evaluation of [11C]4-Methoxy-N-[2-(thiophen-2-yl)imidazo[1,2-a]pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand Selective for the δ-Subunit-Containing γ-Aminobutyric Acid Type A Receptors.
L'Estrade ET, Hansen HD, Falk-Petersen C, Haugaard A, Griem-Krey N, Jung S, Lüddens H, Schirmeister T, Erlandsson M, Ohlsson T, Knudsen GM, Herth MM, Wellendorph P, Frølund B. L'Estrade ET, et al. Among authors: schirmeister t. ACS Omega. 2019 May 22;4(5):8846-8851. doi: 10.1021/acsomega.9b00434. eCollection 2019 May 31. ACS Omega. 2019. PMID: 31459972 Free PMC article.
198 results