Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
5 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Discovery of a Novel Oral Glucocorticoid Receptor Modulator (AZD9567) with Improved Side Effect Profile.
J Med Chem. 2018 Mar 8;61(5):1785-1799. doi: 10.1021/acs.jmedchem.7b01690. Epub 2018 Feb 16.
J Med Chem. 2018.
PMID: 29424542
Discovery of the Oral Leukotriene C4 Synthase Inhibitor (1S,2S)-2-({5-[(5-Chloro-2,4-difluorophenyl)(2-fluoro-2-methylpropyl)amino]-3-methoxypyrazin-2-yl}carbonyl)cyclopropanecarboxylic Acid (AZD9898) as a New Treatment for Asthma.
Munck Af Rosenschöld M, Johannesson P, Nikitidis A, Tyrchan C, Chang HF, Rönn R, Chapman D, Ullah V, Nikitidis G, Glader P, Käck H, Bonn B, Wågberg F, Björkstrand E, Andersson U, Swedin L, Rohman M, Andreasson T, Bergström EL, Jiang F, Zhou XH, Lundqvist AJ, Malmberg A, Ek M, Gordon E, Pettersen A, Ripa L, Davis AM.
Munck Af Rosenschöld M, et al. Among authors: nikitidis a.
J Med Chem. 2019 Sep 12;62(17):7769-7787. doi: 10.1021/acs.jmedchem.9b00555. Epub 2019 Aug 30.
J Med Chem. 2019.
PMID: 31415176
Item in Clipboard
Discovery of AZD8154, a Dual PI3Kγδ Inhibitor for the Treatment of Asthma.
Perry MWD, Björhall K, Bold P, Brűlls M, Börjesson U, Carlsson J, Chang HA, Chen Y, Eriksson A, Fihn BM, Fransson R, Fredlund L, Ge H, Huang H, Karabelas K, Lamm Bergström E, Lever S, Lindmark H, Mogemark M, Nikitidis A, Palmgren AP, Pemberton N, Petersen J, Rodrigo Blomqvist M, Smith RW, Thomas MJ, Ullah V, Tyrchan C, Wennberg T, Westin Eriksson A, Yang W, Zhao S, Öster L.
Perry MWD, et al. Among authors: nikitidis a.
J Med Chem. 2021 Jun 24;64(12):8053-8075. doi: 10.1021/acs.jmedchem.1c00434. Epub 2021 Jun 3.
J Med Chem. 2021.
PMID: 34080862
Item in Clipboard
Surprising lipophilicity observations identify unexpected conformational effects.
Perry MWD, Börjesson U, Nikitidis A, Tyrchan C.
Perry MWD, et al. Among authors: nikitidis a.
Bioorg Med Chem Lett. 2022 Aug 1;69:128786. doi: 10.1016/j.bmcl.2022.128786. Epub 2022 May 12.
Bioorg Med Chem Lett. 2022.
PMID: 35569689
Item in Clipboard
Sequence-based prediction of the intrinsic solubility of peptides containing non-natural amino acids.
Oeller M, Kang RJD, Bolt HL, Gomes Dos Santos AL, Weinmann AL, Nikitidis A, Zlatoidsky P, Su W, Czechtizky W, De Maria L, Sormanni P, Vendruscolo M.
Oeller M, et al. Among authors: nikitidis a.
Nat Commun. 2023 Nov 17;14(1):7475. doi: 10.1038/s41467-023-42940-w.
Nat Commun. 2023.
PMID: 37978172
Free PMC article.
Item in Clipboard
Cite
Cite