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Page 1
Conformational gating, dynamics and allostery in human monoacylglycerol lipase.
Tyukhtenko S, Ma X, Rajarshi G, Karageorgos I, Anderson KW, Hudgens JW, Guo JJ, Nasr ML, Zvonok N, Vemuri K, Wagner G, Makriyannis A. Tyukhtenko S, et al. Among authors: rajarshi g. Sci Rep. 2020 Oct 28;10(1):18531. doi: 10.1038/s41598-020-75497-5. Sci Rep. 2020. PMID: 33116203 Free PMC article.
Synthesis and evaluation of potent and selective MGL inhibitors as a glaucoma treatment.
Alapafuja SO, Malamas MS, Shukla V, Zvonok A, Miller S, Daily L, Rajarshi G, Miyabe CY, Chandrashekhar H, Wood J, Tyukhtenko S, Straiker A, Makriyannis A. Alapafuja SO, et al. Among authors: rajarshi g. Bioorg Med Chem. 2019 Jan 1;27(1):55-64. doi: 10.1016/j.bmc.2018.11.003. Epub 2018 Nov 3. Bioorg Med Chem. 2019. PMID: 30446439 Free PMC article.
Design and Synthesis of Highly Potent and Specific ABHD6 Inhibitors.
Malamas MS, Lamani M, Farah SI, Mohammad KA, Miyabe CY, Rajarshi G, Wu S, Zvonok N, Chandrashekhar H, Wood J, Makriyannis A. Malamas MS, et al. Among authors: rajarshi g. ChemMedChem. 2023 Nov 2;18(21):e202100406. doi: 10.1002/cmdc.202100406. Epub 2021 Sep 6. ChemMedChem. 2023. PMID: 34486233
A comparison of novel, selective fatty acid amide hydrolase (FAAH), monoacyglycerol lipase (MAGL) or dual FAAH/MAGL inhibitors to suppress acute and anticipatory nausea in rat models.
Parker LA, Limebeer CL, Rock EM, Sticht MA, Ward J, Turvey G, Benchama O, Rajarshi G, Wood JT, Alapafuja SO, Makriyannis A. Parker LA, et al. Among authors: rajarshi g. Psychopharmacology (Berl). 2016 Jun;233(12):2265-75. doi: 10.1007/s00213-016-4277-y. Epub 2016 Apr 6. Psychopharmacology (Berl). 2016. PMID: 27048155 Free PMC article.
Design and Structure-Activity Relationships of Isothiocyanates as Potent and Selective N-Acylethanolamine-Hydrolyzing Acid Amidase Inhibitors.
Malamas MS, Pavlopoulos S, Alapafuja SO, Farah SI, Zvonok A, Mohammad KA, West J, Perry NT, Pelekoudas DN, Rajarshi G, Shields C, Chandrashekhar H, Wood J, Makriyannis A. Malamas MS, et al. Among authors: rajarshi g. J Med Chem. 2021 May 13;64(9):5956-5972. doi: 10.1021/acs.jmedchem.1c00076. Epub 2021 Apr 26. J Med Chem. 2021. PMID: 33900772
Probing the carboxyester side chain in controlled deactivation (-)-δ(8)-tetrahydrocannabinols.
Nikas SP, Sharma R, Paronis CA, Kulkarni S, Thakur GA, Hurst D, Wood JT, Gifford RS, Rajarshi G, Liu Y, Raghav JG, Guo JJ, Järbe TU, Reggio PH, Bergman J, Makriyannis A. Nikas SP, et al. Among authors: rajarshi g. J Med Chem. 2015 Jan 22;58(2):665-81. doi: 10.1021/jm501165d. Epub 2014 Dec 16. J Med Chem. 2015. PMID: 25470070 Free PMC article.