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Discovery of a Potent, Selective T-type Calcium Channel Blocker as a Drug Candidate for the Treatment of Generalized Epilepsies.
J Med Chem. 2017 Dec 14;60(23):9769-9789. doi: 10.1021/acs.jmedchem.7b01236. Epub 2017 Nov 20.
J Med Chem. 2017.
PMID: 29116786
Milestones to the Discovery of T-type Calcium Channel Blockers for the Treatment of Generalized Epilepsies.
Bezençon O, Siegrist R, Heidmann B, Pozzi D, Stamm S, Remeň L, Richard S, Simons L, Gaston R, Downing D, Grisostomi C, Roch C, Kessler M, Gatfield J, Moon R, Pfeifer T, Mosbacher J, Reymond I, Ertel EA, de Kanter R, Capeleto B, Fournier E, Rey M, Moccia L, Toeroek-Schafroth M, Roscher R, Schindelholz B.
Bezençon O, et al.
Chimia (Aarau). 2017 Oct 25;71(10):722-729. doi: 10.2533/chimia.2017.722.
Chimia (Aarau). 2017.
PMID: 29070417
Free article.
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Design and synthesis of novel tricyclic benzoxazines as potent 5-HT(1A/B/D) receptor antagonists leading to the discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4H-imidazo[5,1-c][1,4]benzoxazine-3-carboxamide (GSK588045).
Bromidge SM, Arban R, Bertani B, Bison S, Borriello M, Cavanni P, Dal Forno G, Di-Fabio R, Donati D, Fontana S, Gianotti M, Gordon LJ, Granci E, Leslie CP, Moccia L, Pasquarello A, Sartori I, Sava A, Watson JM, Worby A, Zonzini L, Zucchelli V.
Bromidge SM, et al.
J Med Chem. 2010 Aug 12;53(15):5827-43. doi: 10.1021/jm100482n.
J Med Chem. 2010.
PMID: 20590088
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Sarcoidosis with prevalent and severe joint localization: a case report.
Moccia LG, Castaldo S, Sirignano E, Napolitano M, Barra E, Sanduzzi A.
Moccia LG, et al.
Multidiscip Respir Med. 2016 Jun 29;11:27. doi: 10.1186/s40248-016-0064-1. eCollection 2016.
Multidiscip Respir Med. 2016.
PMID: 27358732
Free PMC article.
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Posterior mediastinal extramedullary hematopoiesis secondary to hypoxia.
Solazzo A, D'Auria V, Moccia LG, Vatrella A, Bocchino M, Rea G.
Solazzo A, et al. Among authors: moccia lg.
Transl Med UniSa. 2016 May 16;14:1-4. eCollection 2016 May.
Transl Med UniSa. 2016.
PMID: 27326388
Free PMC article.
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