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Synthesis and Evaluation of Dolastatin 10 Analogues Containing Heteroatoms on the Amino Acid Side Chains.
J Nat Prod. 2017 Sep 22;80(9):2484-2491. doi: 10.1021/acs.jnatprod.7b00359. Epub 2017 Sep 8.
J Nat Prod. 2017.
PMID: 28885014
Investigation of Hydrophilic Auristatin Derivatives for Use in Antibody Drug Conjugates.
Mendelsohn BA, Barnscher SD, Snyder JT, An Z, Dodd JM, Dugal-Tessier J.
Mendelsohn BA, et al. Among authors: barnscher sd.
Bioconjug Chem. 2017 Feb 15;28(2):371-381. doi: 10.1021/acs.bioconjchem.6b00530. Epub 2017 Jan 6.
Bioconjug Chem. 2017.
PMID: 28060485
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Design and Evaluation of ZD06519, a Novel Camptothecin Payload for Antibody Drug Conjugates.
Petersen ME, Brant MG, Lasalle M, Das S, Duan R, Wong J, Ding T, Wu KJ, Siddappa D, Fang C, Zhang W, Wu AML, Hirkala-Schaefer T, Garnett GAE, Fung V, Yang L, Hernandez Rojas A, Lawn SO, Barnscher SD, Rich JR, Colombo R.
Petersen ME, et al. Among authors: barnscher sd.
Mol Cancer Ther. 2024 May 2;23(5):606-618. doi: 10.1158/1535-7163.MCT-23-0822.
Mol Cancer Ther. 2024.
PMID: 38354417
Free PMC article.
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Structure-Activity Relationships of Bis-Intercalating Peptides and Their Application as Antibody-Drug Conjugate Payloads.
Petersen ME, Brant MG, Lasalle M, Fung VKC, Rojas AH, Wong J, Das S, Barnscher SD, Rich JR, Winters GC.
Petersen ME, et al. Among authors: barnscher sd.
J Med Chem. 2023 Jun 22;66(12):8288-8309. doi: 10.1021/acs.jmedchem.3c00760. Epub 2023 Jun 12.
J Med Chem. 2023.
PMID: 37307297
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Generation and structure-activity relationships of novel imidazo-thienopyridine based TLR7 agonists: application as payloads for immunostimulatory antibody drug-conjugates.
Brant MG, Garnett GAE, Guedia J, Lasalle M, Lawn S, Petersen ME, Duan R, Mendez-Campos J, Hirkala-Schaefer T, Winters GC, Barnscher SD.
Brant MG, et al. Among authors: barnscher sd.
Bioorg Med Chem Lett. 2023 Jul 15;91:129348. doi: 10.1016/j.bmcl.2023.129348. Epub 2023 May 20.
Bioorg Med Chem Lett. 2023.
PMID: 37217025
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